SCHEMBL7857530

SCHEMBL7857530

Cc1noc(NS(=O)(=O)c2ccc(Cl)cc2)c1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 18/20 1.00
EDNRB P24530 13/20 1.00
MEN1 O00255 1/20 0.74
CYP2C9 P11712 1/20 0.74
TSHR P16473 1/20 0.74
CYP2C19 P33261 1/20 0.74
ADRA1A P35348 1/20 0.74
KMT2A Q03164 1/20 0.74
P2RY1 P47900 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7857604 0.86 EDNRA (0.76) EDNRAEDNRBMEN1CYP2C9TSHR
SCHEMBL7222860 0.85 EDNRA (1.00) EDNRAEDNRB
SCHEMBL7860467 0.85 EDNRA (1.00) EDNRAEDNRBMEN1CYP2C9TSHR
SCHEMBL7856711 0.85 EDNRA (1.00) EDNRAEDNRBMEN1CYP2C9TSHR
Sulfisoxazole SCHEMBL23467 0.85 EDNRA (1.00) EDNRAEDNRBMEN1CYP2C9TSHR
SCHEMBL7849834 0.85 EDNRA (0.78) EDNRAEDNRBMEN1CYP2C9TSHR
Sulfisoxazole SCHEMBL788644 0.85 EDNRA (1.00) EDNRAEDNRBMEN1CYP2C9TSHR
SCHEMBL7716850 0.84 EDNRA (1.00) EDNRAEDNRBMEN1CYP2C9TSHR
SCHEMBL7857285 0.84 EDNRA (1.00) EDNRAEDNRBMEN1CYP2C9TSHR
Sulfisoxazole SCHEMBL5917298 0.84 EDNRA (0.97) EDNRAEDNRBMEN1CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1069114-A2 Sulfonamides and derivatives thereof that modulate the activity of endothelin TEXAS BIOTECHNOLOGY CORPORATION (US) 2001-01-17 EP disclosed