SCHEMBL78590

SCHEMBL78590

CC(C)(C)c1cc(CNC(=O)C2CC2)ccc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 4/20 0.54
P2RX7 Q99572 5/20 0.51
ERCC1 P07992 1/20 0.50
ERCC4 Q92889 1/20 0.50
ALDH1A1 P00352 3/20 0.49
HPGD P15428 2/20 0.49
KDM4E B2RXH2 1/20 0.49
ALOX15 P16050 1/20 0.49
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
SLC13A5 Q86YT5 1/20 0.46
NPC1 O15118 1/20 0.46
PKM P14618 1/20 0.46
RAB9A P51151 1/20 0.46
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
USP2 O75604 1/20 0.44
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1751211 0.83 EPHX2 (0.48) EPHX2P2RX7ERCC1ERCC4ALDH1A1
SCHEMBL30791545 0.83 EPHX2 (0.61) EPHX2P2RX7ERCC1ERCC4ALDH1A1
SCHEMBL91263 0.81 ERCC1 (0.52) EPHX2P2RX7ERCC1ERCC4ALDH1A1
SCHEMBL2635463 0.80 ERCC1 (0.55) EPHX2ERCC1ERCC4ALDH1A1HPGD
SCHEMBL13190006 0.79 ERCC1 (0.54) EPHX2P2RX7ERCC1ERCC4ALDH1A1
SCHEMBL1750644 0.79 ERCC1 (0.54) EPHX2P2RX7ERCC1ERCC4ALDH1A1
SCHEMBL4004065 0.79 ERCC1 (0.54) EPHX2P2RX7ERCC1ERCC4ALDH1A1
SCHEMBL30491752 0.78 ERCC1 (0.52) EPHX2ERCC1ERCC4ALDH1A1HPGD
SCHEMBL14782772 0.78 ERCC1 (0.52) EPHX2ERCC1ERCC4ALDH1A1HPGD
SCHEMBL14782977 0.77 HPGD (0.55) EPHX2P2RX7ERCC1ERCC4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed