SCHEMBL7859779

SCHEMBL7859779

COc1cc2c(C3CCNCC3)c[nH]c2cc1F

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
APP P05067 6/20 0.51
HTR2C P28335 4/20 0.48
ADRB2 P07550 1/20 0.48
HTR6 P50406 1/20 0.47
HTR1A P08908 4/20 0.46
MTNR1A P48039 1/20 0.46
MTNR1B P49286 1/20 0.46
HTR2B P41595 1/20 0.42
NMT2 O60551 1/20 0.41
NMT1 P30419 1/20 0.41
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL8818387 0.84 APP (0.54) APPHTR1ASLC6A4
SCHEMBL5374013 0.84 APP (0.58) APPHTR1ASLC6A4
SCHEMBL22491588 0.79 APP (0.54) APPHTR2CADRB2HTR6NMT2
SCHEMBL19702109 0.76 HTR2C (0.51) HTR2CHTR6HTR1ASLC6A2SLC6A4
SCHEMBL8317118 0.75 HTR2C (0.57) APPHTR2CADRB2HTR6MTNR1A
SCHEMBL2264043 0.75 HTR2C (0.60) APPHTR2CADRB2HTR6HTR1A
SCHEMBL7866276 0.75 HTR2C (0.44) HTR2CHTR6HTR1ASLC6A2SLC6A4
Hydrochloric Acid SCHEMBL11841895 0.74 HTR2C (0.58) APPHTR2CADRB2HTR6HTR2B
Hydrochloric Acid SCHEMBL11847902 0.74 HTR2C (0.59) APPHTR2CADRB2HTR6HTR1A
SCHEMBL2781509 0.73 HTR2C (0.62) APPHTR2CADRB2HTR6HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077213-A2 Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 2001-02-21 EP disclosed
US-6046215-A A PIPERIDINYLBENZOTHIOPHENES USEFUL FOR TRATING BRAIN DISORDERS ELI LILLY AND COMPANY (US) 2000-04-04 US disclosed
US-5846982-A Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 1998-12-08 US disclosed
EP-0812826-A1 1H-indole and benzo(b)thiophene derivatives with 4-(1,2,3,6-tetra:hydro:pyridinyl)- and 4-piperidinyl-groups bound to the heterocyclic ring as inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1997-12-17 EP disclosed