SCHEMBL7861249

SCHEMBL7861249

CCN(CC)Cc1cccc(-c2nc3c(OC(=O)O)cccc3[nH]2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.53
DHODH Q02127 3/20 0.44
VSIR Q9H7M9 3/20 0.43
MMP2 P08253 2/20 0.43
MMP9 P14780 2/20 0.43
MMP8 P22894 2/20 0.43
CHEK1 O14757 1/20 0.43
MAP4K4 O95819 1/20 0.43
LCK P06239 1/20 0.43
CSF1R P07333 1/20 0.43
PIM1 P11309 1/20 0.43
PHKG2 P15735 1/20 0.43
MARK3 P27448 1/20 0.43
KDR P35968 1/20 0.43
FLT3 P36888 1/20 0.43
CLK2 P49760 1/20 0.43
GSK3A P49840 1/20 0.43
ITK Q08881 1/20 0.43
MAP4K2 Q12851 1/20 0.43
DYRK1A Q13627 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6379926 0.91 PARP1 (0.58) PARP1VSIRCHEK1MAP4K4LCK
SCHEMBL7859132 0.89 PARP1 (0.52) PARP1DHODHCHEK1MAP4K4LCK
SCHEMBL7138597 0.81 PARP1 (0.80) PARP1DHODHCHEK1MAP4K4LCK
SCHEMBL6383270 0.81 PARP1 (0.51) PARP1VSIRCHEK1MAP4K4LCK
SCHEMBL6380476 0.80 PARP1 (0.72) PARP1VSIRMAP4K4PIM1PIM3
SCHEMBL6379799 0.80 PARP1 (0.56) PARP1DHODHCHEK1MAP4K4LCK
SCHEMBL7853256 0.78 PARP1 (0.65) PARP1DHODHHPSE
SCHEMBL7860364 0.78 PARP1 (0.69) PARP1DHODHKDRAURKB
SCHEMBL6383675 0.75 PARP1 (0.57) PARP1DHODHVSIRPIM1PIM3
SCHEMBL6381528 0.74 PARP1 (0.58) PARP1VSIRMAP4K4PIM1PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131301-A1 2-PHENYLBENZIMIDAZOLES AND 2-PHENYLINDOLES, AND PRODUCTION AND USE THEREOF BASF AKTIENGESELLSCHAFT (DE) 2001-09-12 EP disclosed
WO-2000029384-A1 2-PHENYLBENZIMIDAZOLES AND 2-PHENYLINDOLES, AND PRODUCTION AND USE THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-05-25 WO disclosed