SCHEMBL7861970

SCHEMBL7861970

N=C(N)Nc1cccc(C(=O)Nc2cccc(CCC(=O)O)c2)c1

nearest known ligand 0.76

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 4/20 0.76
ITGA2B P08514 4/20 0.76
ITGAV P06756 2/20 0.55
ITGB1 P05556 1/20 0.55
ITGB5 P18084 1/20 0.55
NR1H4 Q96RI1 6/20 0.52
PPARD Q03181 3/20 0.52
PPARG P37231 2/20 0.52
PPARA Q07869 2/20 0.52
SIRT1 Q96EB6 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.49
HSPH1 Q92598 1/20 0.48
ALDH1A1 P00352 1/20 0.47
HPSE Q9Y251 1/20 0.47
KMT2A Q03164 1/20 0.47
KCNK3 O14649 1/20 0.47
KCNK9 Q9NPC2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7373419 0.91 ITGB3 (0.66) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7457414 0.90 ITGB3 (0.84) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7346500 0.89 ITGB3 (0.60) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL8371218 0.89 ITGB3 (0.61) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL8500653 0.88 ITGB3 (0.60) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7856521 0.88 PPARG (0.60) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7864209 0.87 HPSE (0.62) ITGB3ITGA2BNR1H4PPARDPPARG
SCHEMBL7378120 0.86 ITGB3 (0.57) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7856482 0.86 ITGB3 (0.65) ITGB3ITGA2BITGB1NR1H4PPARD
SCHEMBL7380122 0.85 ITGB3 (0.56) ITGB3ITGA2BITGAVITGB1ITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP claimed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP disclosed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO disclosed