SCHEMBL7862288

SCHEMBL7862288

CCc1c(C(=O)N2CCOc3ccc(C4=NNC(=O)C4)cc3C2)ccc(S(C)(=O)=O)c1F

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 1/20 0.55
PIK3CA P42336 15/20 0.55
PDE3B Q13370 2/20 0.39
PDE3A Q14432 2/20 0.39
RIPK1 Q13546 1/20 0.39
CREBBP Q92793 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7859563 0.85 PRKDC (0.61) PRKDCPIK3CARIPK1CREBBP
SCHEMBL3754519 0.85 PRKDC (0.62) PRKDCPIK3CARIPK1
SCHEMBL3749989 0.84 PRKDC (0.61) PRKDCPIK3CARIPK1
SCHEMBL3748164 0.83 PRKDC (0.57) PRKDCPIK3CARIPK1
SCHEMBL3757923 0.83 PRKDC (0.55) PRKDCPIK3CARIPK1
SCHEMBL3762511 0.83 PRKDC (0.60) PRKDCPIK3CARIPK1CREBBP
SCHEMBL3756142 0.83 PIK3CA (0.60) PRKDCPIK3CARIPK1CREBBP
SCHEMBL3755006 0.83 PRKDC (0.64) PRKDCPIK3CARIPK1CREBBP
SCHEMBL3750661 0.83 PRKDC (0.66) PRKDCPIK3CARIPK1
SCHEMBL3718769 0.83 PRKDC (0.59) PRKDCPIK3CARIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118208-A1 BENZOXAZEPIN-4- (5H) -YL DERIVATIVES AND THEIR USE TO TREAT CANCER EXELIXIS, INC. (US) 2010-10-14 WO disclosed