SCHEMBL7862423

SCHEMBL7862423

CCCCCC(O)(CO)Cn1cncn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.45
ALDH1A1 P00352 1/20 0.45
FDPS P14324 1/20 0.43
HSP90AA1 P07900 2/20 0.41
CYP2C9 P11712 3/20 0.39
CYP2C19 P33261 3/20 0.39
LMNA P02545 2/20 0.39
CYP19A1 P11511 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
ADRA1A P35348 1/20 0.39
CYP51A1 Q16850 1/20 0.39
KMT2A Q03164 1/20 0.35
EGLN3 Q9H6Z9 1/20 0.33
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
TLR8 Q9NR97 1/20 0.30
TLR7 Q9NYK1 1/20 0.30
CYP2B6 P20813 1/20 0.30
CYP3A5 P20815 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10819000 0.92 FDPS (0.46) CYP3A4ALDH1A1FDPSHSP90AA1CYP2C9
SCHEMBL9010566 0.89 FDPS (0.44) CYP3A4ALDH1A1FDPSHSP90AA1CYP2C9
SCHEMBL10816070 0.87 FDPS (0.42) CYP3A4ALDH1A1FDPSHSP90AA1CYP2C9
SCHEMBL11083531 0.87 FDPS (0.45) CYP3A4ALDH1A1FDPSHSP90AA1CYP2C9
SCHEMBL9770713 0.83 CYP3A4 (0.59) CYP3A4ALDH1A1FDPSHSP90AA1CYP2C9
SCHEMBL8800253 0.83 FDPS (0.39) CYP3A4ALDH1A1FDPSHSP90AA1CYP2C9
SCHEMBL9863651 0.82 FDPS (0.44) CYP3A4ALDH1A1FDPSHSP90AA1CYP2C9
SCHEMBL9770830 0.82 CYP3A4 (0.58) CYP3A4ALDH1A1FDPSHSP90AA1CYP2C9
SCHEMBL9770607 0.82 CYP3A4 (0.58) CYP3A4ALDH1A1FDPSHSP90AA1CYP2C9
SCHEMBL9770734 0.78 CYP3A4 (0.48) CYP3A4ALDH1A1FDPSHSP90AA1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1120397-A2 Process for preparing triazole derivative KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 2001-08-01 EP disclosed
US-6046354-A CHEMICAL INTERMEDIATES, E.G. 2-ARYL-1,3-DIACYLOXY-2-PROPANOL, FOR DRUGS AND FUNGICIDES,E.G. (R)-2-(2,4-DIFLUOROPHENYL)-3-(1H-1,2,4-TRIAZOLE-1-YL)-PROPANE-1,2-DIOL, KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 2000-04-04 US disclosed
US-5840553-A OPTICALLY ACTIVE 2-ARYL-3-ACYLOXY-1,2,-PROPANE DIOL USING A MICROORGANISM OR ENZYME DERIVED FROM PORCINE PANCREAS; VIA STEREOSPECIFIC HYDROLYSIS OF A 2-ARYL-1,3-DIACYLOXY-2-PROPANOL; SYNTHETIC CHEMICAL INTERMEDIATES, FUNGICIDES KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1998-11-24 US disclosed
US-5654472-A OPTICALLY PURE 2-ARYL-3-ACYLOXY-1,2-PROPANEDIOL COMPOUNDS; CHEMICAL INTERMEDIATES KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1997-08-05 US disclosed
EP-0704419-A1 PROCESS FOR PRODUCING TRIAZOLE DERIVATIVE KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1996-04-03 EP disclosed