SCHEMBL7863950

SCHEMBL7863950

Cc1c(Cl)cc(C(=O)O)c(Cl)c1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.44
TSHR P16473 3/20 0.42
ALDH1A1 P00352 3/20 0.42
TP53 P04637 1/20 0.42
CASP1 P29466 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
AKR1C2 P52895 2/20 0.41
AKR1C1 Q04828 2/20 0.41
AKR1C3 P42330 2/20 0.41
AKR1C4 P17516 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
MYC P01106 1/20 0.41
NR4A1 P22736 1/20 0.41
CTSB P07858 1/20 0.41
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
KDM4E B2RXH2 2/20 0.40
MAPT P10636 2/20 0.40
HPGD P15428 2/20 0.40
PKM P14618 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8333633 0.87 CYP3A4 (0.44) CYP3A4TSHRALDH1A1TP53CASP1
SCHEMBL27675106 0.84 TDP1 (0.45) CYP3A4TSHRALDH1A1TP53CASP1
SCHEMBL28217274 0.84 MEN1 (0.45) CYP3A4TSHRALDH1A1TP53CASP1
SCHEMBL28137972 0.83 CYP3A4 (0.41) CYP3A4TSHRALDH1A1TP53CASP1
SCHEMBL11231441 0.83 MYC (0.42) CYP3A4TSHRALDH1A1TP53CASP1
SCHEMBL7863941 0.83 MEN1 (0.44) CYP3A4TSHRALDH1A1TP53CASP1
SCHEMBL10630705 0.82 NOTUM (0.42) CYP3A4TSHRALDH1A1TP53CASP1
SCHEMBL10625931 0.82 CYP3A4 (0.48) CYP3A4TSHRALDH1A1TP53CASP1
SCHEMBL4314431 0.79 KDM4E (0.50) CYP3A4TSHRALDH1A1TP53CASP1
SCHEMBL2149302 0.79 AKR1C2 (0.52) TSHRALDH1A1TP53CASP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9238657-B2 Cephalosporin having catechol group SHIONOGI & CO., LTD. (JP) 2016-01-19 US disclosed
US-20110190254-A1 CEPHALOSPORIN HAVING CATECHOL GROUP SHIONOGI & CO., LTD. (JP) 2011-08-04 US disclosed
WO-2001083420-A2 METHOD OF MAKING SUBSTITUTED DIHALO AROMATIC ACID CHLORIDES OCCIDENTAL CHEMICAL CORPORATION (US) 2001-11-08 WO disclosed
US-6303812-B1 ADDING WATER TO A MIXTURE CONTAINING A CUPROUS HALIDE, CUPROUS ACETATE OR PROPIONATE, AND CERTAIN DEHALOGENATED AROMATIC PRODUCTS, SUCH AS METHYL 3,5-DICHLORO-4-METHYLBENZOATE, CAUSES THE MIXTURE TO SEPARATE INTO ORGANIC AND AQUEOUS PHASES OCCIDENTAL CHEMICAL CORPORATION 2001-10-16 US disclosed
US-6118018-A Chlorination and bromination of aromatic compounds at atmospheric pressure OCCIDENTAL CHEMICAL CORPORATION (US) 2000-09-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110190254-A1 CEPHALOSPORIN HAVING CATECHOL GROUP NRDC, LUC7L2, NR0B1 CYP3A4 1037/4885TSHR 2183/4885ALDH1A1 2808/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.