SCHEMBL7863941

SCHEMBL7863941

Cc1c(Cl)cc(C(=O)O)c(C)c1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
TDP1 Q9NUW8 2/20 0.44
KDM4E B2RXH2 2/20 0.44
TSHR P16473 3/20 0.42
ALDH1A1 P00352 3/20 0.42
TP53 P04637 1/20 0.42
CASP1 P29466 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
AKR1C2 P52895 2/20 0.41
AKR1C1 Q04828 2/20 0.41
AKR1C3 P42330 2/20 0.41
AKR1C4 P17516 1/20 0.41
MYC P01106 1/20 0.41
NR4A1 P22736 1/20 0.41
CTSB P07858 1/20 0.41
MAPT P10636 2/20 0.40
HPGD P15428 2/20 0.40
PKM P14618 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8333633 0.87 CYP3A4 (0.44) MEN1KMT2ATDP1KDM4ETSHR
SCHEMBL28217274 0.84 MEN1 (0.45) MEN1KMT2ATDP1KDM4ETSHR
SCHEMBL691741 0.83 AKR1C2 (0.52) MEN1KMT2ATDP1KDM4ETSHR
SCHEMBL2149302 0.83 AKR1C2 (0.52) MEN1KMT2ATDP1KDM4ETSHR
SCHEMBL11343587 0.83 ALDH1A1 (0.40) MEN1KMT2ATDP1KDM4ETSHR
SCHEMBL7863950 0.83 CYP3A4 (0.44) MEN1KMT2ATDP1KDM4ETSHR
SCHEMBL11181385 0.83 KDM4E (0.44) MEN1KMT2ATDP1KDM4ETSHR
SCHEMBL23513273 0.82 NOTUM (0.42) MEN1KMT2ATDP1KDM4ETSHR
SCHEMBL10354535 0.82 KDM4E (0.48) MEN1KMT2ATDP1KDM4ETSHR
SCHEMBL27281805 0.82 KDM4E (0.48) MEN1KMT2ATDP1KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303812-B1 ADDING WATER TO A MIXTURE CONTAINING A CUPROUS HALIDE, CUPROUS ACETATE OR PROPIONATE, AND CERTAIN DEHALOGENATED AROMATIC PRODUCTS, SUCH AS METHYL 3,5-DICHLORO-4-METHYLBENZOATE, CAUSES THE MIXTURE TO SEPARATE INTO ORGANIC AND AQUEOUS PHASES OCCIDENTAL CHEMICAL CORPORATION 2001-10-16 US claimed
US-6201152-B1 HEATING MIXTURE OF METHYL-3,5-DICHLORO-4-METHYLBENZOATE AND ALPHA,ALPHA,ALPHA-TRICHLOROMETHYLBENZENE IN PRESENCE OF AMMONIUM MOLYBDATE CATALYST OCCIDENTAL CHEMICAL CORPORATION 2001-03-13 US claimed
WO-2001083420-A2 METHOD OF MAKING SUBSTITUTED DIHALO AROMATIC ACID CHLORIDES OCCIDENTAL CHEMICAL CORPORATION (US) 2001-11-08 WO disclosed
US-6303812-B1 ADDING WATER TO A MIXTURE CONTAINING A CUPROUS HALIDE, CUPROUS ACETATE OR PROPIONATE, AND CERTAIN DEHALOGENATED AROMATIC PRODUCTS, SUCH AS METHYL 3,5-DICHLORO-4-METHYLBENZOATE, CAUSES THE MIXTURE TO SEPARATE INTO ORGANIC AND AQUEOUS PHASES OCCIDENTAL CHEMICAL CORPORATION 2001-10-16 US disclosed
US-6201152-B1 HEATING MIXTURE OF METHYL-3,5-DICHLORO-4-METHYLBENZOATE AND ALPHA,ALPHA,ALPHA-TRICHLOROMETHYLBENZENE IN PRESENCE OF AMMONIUM MOLYBDATE CATALYST OCCIDENTAL CHEMICAL CORPORATION 2001-03-13 US disclosed
US-6201152-B1 HEATING MIXTURE OF METHYL-3,5-DICHLORO-4-METHYLBENZOATE AND ALPHA,ALPHA,ALPHA-TRICHLOROMETHYLBENZENE IN PRESENCE OF AMMONIUM MOLYBDATE CATALYST OCCIDENTAL CHEMICAL CORPORATION 2001-03-13 US disclosed
US-6118018-A Chlorination and bromination of aromatic compounds at atmospheric pressure OCCIDENTAL CHEMICAL CORPORATION (US) 2000-09-12 US disclosed