SCHEMBL7864258

SCHEMBL7864258

C=C(C)OC(=O)NC1(C(=O)N[C@@H](Cc2ccc(-c3ccc(S(=O)(=O)C(C)C)cc3)cc2)C(N)=O)CCOCC1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 13/20 0.40
ITGA4 P13612 13/20 0.40
ITGB7 P26010 8/20 0.40
CTSC P53634 2/20 0.37
ECE1 P42892 1/20 0.34
TACR2 P21452 1/20 0.34
MMP1 P03956 2/20 0.34
MMP13 P45452 2/20 0.34
MMP2 P08253 1/20 0.34
MMP3 P08254 1/20 0.34
MMP9 P14780 1/20 0.34
MMP8 P22894 1/20 0.34
MMP14 P50281 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL300140 0.87 ITGB1 (0.42) ITGB1ITGA4ITGB7CTSC
SCHEMBL300141 0.87 ITGB1 (0.42) ITGB1ITGA4ITGB7CTSC
SCHEMBL9888300 0.85 CTSC (0.49) ITGB1ITGA4CTSCTACR2MMP1
SCHEMBL9888327 0.80 F11 (0.35) ITGB1ITGA4ITGB7
SCHEMBL9888289 0.79 CTSC (0.37) ITGB1ITGA4ITGB7CTSCECE1
SCHEMBL9888321 0.79 CTSC (0.54) CTSCTACR2
SCHEMBL2892835 0.78 ITGB1 (0.41) ITGB1ITGA4ITGB7CTSCTACR2
SCHEMBL2892834 0.78 ITGB1 (0.41) ITGB1ITGA4ITGB7CTSCTACR2
SCHEMBL298671 0.77 ITGB1 (0.44) ITGB1ITGA4ITGB7CTSCECE1
SCHEMBL9888277 0.76 CTSC (0.40) CTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010128324-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 WO disclosed