SCHEMBL7864439

SCHEMBL7864439

Clc1cccc(-c2nnc([C@@H]3CCCNC3)n2C2CC2)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 5/20 0.40
OPRM1 P35372 2/20 0.37
OPRD1 P41143 2/20 0.37
OPRK1 P41145 2/20 0.37
OPRL1 P41146 2/20 0.37
CHRM1 P11229 1/20 0.35
HRH1 P35367 1/20 0.35
SLC6A2 P23975 3/20 0.35
SLC6A4 P31645 3/20 0.35
SLC6A3 Q01959 3/20 0.35
CYP2D6 P10635 2/20 0.35
KCNH2 Q12809 2/20 0.35
CNR2 P34972 1/20 0.35
HTR3E A5X5Y0 1/20 0.35
HTR3B O95264 1/20 0.35
HTR2B P41595 1/20 0.35
HTR3A P46098 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
HTR3D Q70Z44 1/20 0.35
HTR3C Q8WXA8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL555729 0.74 REN (0.41) P2RX7KCNH2
Hydrochloric Acid SCHEMBL557460 0.73 REN (0.41) KCNH2
SCHEMBL7347495 0.67 KCNH2 (0.51) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL17103013 0.64 CYP2D6 (0.53) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL10810726 0.63 CYP2D6 (0.39) CHRM1HRH1SLC6A2SLC6A4SLC6A3
SCHEMBL3697519 0.63 HTR2A (0.51) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
Hydrochloric Acid SCHEMBL2884606 0.62 HTR2A (0.50) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL25044088 0.61 SLC6A2 (0.45) OPRL1SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL16110833 0.61 HTR2A (0.47) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL1914524 0.61 MAPK1 (0.45) CHRM1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed