SCHEMBL7865237

SCHEMBL7865237

O=C(NC1CCCCNC1)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 5/20 0.55
MAPK1 P28482 1/20 0.54
OPRK1 P41145 1/20 0.54
NPC1 O15118 5/20 0.54
RAB9A P51151 5/20 0.54
PKM P14618 1/20 0.51
CDK2AP1 O14519 1/20 0.50
HDAC4 P56524 1/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
GRM5 P41594 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1163022 0.95 MAPK1 (0.59) CHEK1MAPK1OPRK1NPC1RAB9A
SCHEMBL28280152 0.95 MAPK1 (0.59) CHEK1MAPK1OPRK1NPC1RAB9A
SCHEMBL1163023 0.95 MAPK1 (0.59) CHEK1MAPK1OPRK1NPC1RAB9A
SCHEMBL1250846 0.89 MEN1 (0.54) MAPK1OPRK1NPC1RAB9AHDAC4
SCHEMBL5230051 0.89 MEN1 (0.54) MAPK1OPRK1NPC1RAB9AHDAC4
SCHEMBL8491815 0.89 MEN1 (0.54) MAPK1OPRK1NPC1RAB9AHDAC4
Hydrochloric Acid SCHEMBL28156652 0.88 MEN1 (0.53) MAPK1OPRK1NPC1RAB9AHDAC4
Hydrochloric Acid SCHEMBL994487 0.88 MEN1 (0.53) MAPK1OPRK1NPC1RAB9AHDAC4
Hydrochloric Acid SCHEMBL28155972 0.88 MEN1 (0.53) MAPK1OPRK1NPC1RAB9AHDAC4
Cadaverine Tartrate SCHEMBL28008723 0.88 MAPK1 (0.52) CHEK1MAPK1OPRK1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1085888-A1 MULTIVALENT AGONISTS, PARTIAL AGONISTS, INVERSE AGONISTS AND ANTAGONISTS OF THE 5-HT 3? RECEPTORS Advanced Medicine, Inc. (US) 2001-03-28 EP disclosed
WO-1999064046-A9 MULTIVALENT AGONISTS, PARTIAL AGONISTS, INVERSE AGONISTS AND ANTAGONISTS OF THE 5-HT3 RECEPTORS ADVANCED MEDICINE INC (US) 2000-04-20 WO disclosed
WO-1999064046-A1 MULTIVALENT AGONISTS, PARTIAL AGONISTS, INVERSE AGONISTS AND ANTAGONISTS OF THE 5-HT3 RECEPTORS ADVANCED MEDICINE, INC. (US) 1999-12-16 WO disclosed