SCHEMBL7867942

SCHEMBL7867942

CS(=O)(=O)c1nccc(-n2ccc3ccccc32)n1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 9/20 0.58
CDC7 O00311 8/20 0.58
ROCK1 Q13464 6/20 0.58
MKNK1 Q9BUB5 3/20 0.45
MAPK8 P45983 2/20 0.45
MAPK9 P45984 2/20 0.45
MKNK2 Q9HBH9 2/20 0.45
MAPK10 P53779 1/20 0.45
JUN P05412 1/20 0.42
RPS6KA5 O75582 1/20 0.40
MAPT P10636 1/20 0.40
PRKD3 O94806 1/20 0.39
PRKCG P05129 1/20 0.39
PRKCB P05771 1/20 0.39
PRKCA P17252 1/20 0.39
PRKACA P17612 1/20 0.39
PRKACG P22612 1/20 0.39
PRKACB P22694 1/20 0.39
PRKCH P24723 1/20 0.39
PRKCI P41743 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7022083 0.79 ROCK1 (0.59) ROCK1MKNK1MKNK2
SCHEMBL19533417 0.77 CDK2 (0.67) CDK2CDC7ROCK1MKNK1MAPK8
SCHEMBL3823223 0.76 CDK1 (0.53) CDK2MKNK1MAPK8MAPK9MKNK2
SCHEMBL6301371 0.75 KDR (0.55)
SCHEMBL5102168 0.75 CDK2 (0.63) CDK2CDC7ROCK1MKNK1MAPK8
SCHEMBL5659028 0.74 RPS6KA5 (0.68) CDK2CDC7ROCK1MKNK1MAPK8
SCHEMBL30753972 0.74 CDC7 (1.00) CDK2CDC7ROCK1MAP3K14
SCHEMBL9377410 0.74 CDC7 (1.00) CDK2CDC7ROCK1MAP3K14
SCHEMBL30459871 0.74 RPS6KA5 (0.68) CDK2CDC7ROCK1MKNK1MAPK8
SCHEMBL17918815 0.73 BRAF (0.38) ROCK1MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316444-B1 SRC kinase inhibitor compounds MERCK & CO., INC. 2001-11-13 US disclosed