SCHEMBL7868054

SCHEMBL7868054

C=C(C)OC(=O)NC1(C(=O)N[C@H](C#N)Cc2ccc(-c3cccc(C#N)c3)cc2)CCOCC1

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSC P53634 19/20 0.53
KCNH2 Q12809 3/20 0.53
LTB4R Q15722 1/20 0.53
LTB4R2 Q9NPC1 1/20 0.53
CTSK P43235 1/20 0.45
MME P08473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2892625 0.88 CTSC (0.54) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL2892624 0.88 CTSC (0.54) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL2884861 0.86 CTSC (0.61) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL9888300 0.82 CTSC (0.49) CTSCKCNH2LTB4RLTB4R2
SCHEMBL9888342 0.82 CTSC (0.50) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL2889502 0.80 CTSC (0.81) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL2889507 0.80 CTSC (0.81) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL2889383 0.79 CTSC (0.64) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL2889385 0.79 CTSC (0.64) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL7871672 0.77 CTSS (0.44) CTSCKCNH2LTB4RLTB4R2CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010128324-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 WO disclosed