SCHEMBL7868902

SCHEMBL7868902

COc1ccc(S(=O)(=O)CC(NC(=O)CN(C(=O)CNC(=O)OC(C)(C)C)c2ccccc2)C(=O)NO)cc1

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 17/20 0.59
MMP9 P14780 4/20 0.40
MMP1 P03956 4/20 0.38
MMP2 P08253 1/20 0.38
MMP7 P09237 1/20 0.38
MMP12 P39900 1/20 0.38
BMP1 P13497 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7866993 0.93 MMP13 (0.48) MMP13MMP9MMP1MMP2BMP1
SCHEMBL7870727 0.89 MMP13 (0.60) MMP13MMP9MMP1MMP2MMP12
SCHEMBL7868903 0.87 MMP13 (0.56) MMP13MMP9MMP1MMP2BMP1
SCHEMBL7874056 0.85 MMP13 (0.64) MMP13MMP9MMP1MMP2MMP7
Trifluoroacetic Acid SCHEMBL7862145 0.84 MMP13 (0.51) MMP13MMP9MMP1MMP2BMP1
SCHEMBL7870766 0.81 MMP13 (0.48) MMP13MMP9MMP2BMP1
SCHEMBL7868827 0.79 MMP13 (0.78) MMP13MMP9MMP1MMP2MMP7
SCHEMBL7866994 0.79 MMP13 (0.45) MMP13MMP9MMP2
SCHEMBL7867020 0.78 MMP13 (0.53) MMP13MMP9MMP1MMP2
SCHEMBL7866976 0.77 MMP13 (0.44) MMP13MMP9MMP1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0994104-A1 ARYL (SULFIDE, SULFOXIDE AND SULFONE) DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2000-04-19 EP claimed
US-6300514-B1 INHIBITING MATRIX METALLOPROTEINASES ONO PHARMACEUTICAL CO., LTD. (JP) 2001-10-09 US disclosed
EP-0994104-A1 ARYL (SULFIDE, SULFOXIDE AND SULFONE) DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2000-04-19 EP disclosed