SCHEMBL7868917

SCHEMBL7868917

Cc1ccc(-c2ccccc2)c(C(=O)N2C[C@@H]3C[C@@H]3CC2COc2ccc(C(F)(F)F)nn2)n1

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 11/20 0.52
HCRTR1 O43613 14/20 0.50
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL609531 1.00 HCRTR2 (0.52) HCRTR2HCRTR1CYP3A4
SCHEMBL609329 0.90 HCRTR2 (0.64) HCRTR2HCRTR1
SCHEMBL7869499 0.87 CYP3A4 (0.54) HCRTR2HCRTR1CYP3A4
SCHEMBL610097 0.87 CYP3A4 (0.54) HCRTR2HCRTR1CYP3A4
SCHEMBL607593 0.87 HCRTR2 (0.50) HCRTR2HCRTR1
SCHEMBL7869493 0.87 HCRTR2 (0.50) HCRTR2HCRTR1
SCHEMBL611279 0.84 CYP3A4 (0.52) HCRTR2HCRTR1CYP3A4
SCHEMBL7869957 0.83 HCRTR1 (0.45) HCRTR2HCRTR1CYP3A4
SCHEMBL609528 0.83 HCRTR1 (0.45) HCRTR2HCRTR1CYP3A4
SCHEMBL7861581 0.81 HCRTR1 (0.42) HCRTR2HCRTR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010122151-A1 3 -AZABICYCLO [4.1.0] HEPTANES USED AS OREXIN ANTAGONISTS GLAXO GROUP LIMITED (GB) 2010-10-28 WO disclosed