SCHEMBL7869103

SCHEMBL7869103

CCCS(=O)(=O)Nc1cccc(C(=O)c2c[nH]c3ncc(/C(C=N)=C/NC)cc23)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 5/20 0.49
CYP2C9 P11712 8/20 0.46
RIPK2 O43353 2/20 0.46
RAF1 P04049 2/20 0.46
KDR P35968 2/20 0.46
MAP2K2 P36507 2/20 0.46
TGFBR2 P37173 2/20 0.46
NEK2 P51955 2/20 0.46
MAP2K1 Q02750 2/20 0.46
TNK2 Q07912 2/20 0.46
MAP2K5 Q13163 2/20 0.46
PTK6 Q13882 2/20 0.46
NEK11 Q8NG66 2/20 0.46
MAP3K20 Q9NYL2 2/20 0.46
MAP4K5 Q9Y4K4 2/20 0.46
BMPR1B O00238 1/20 0.46
PLK4 O00444 1/20 0.46
PIR O00625 1/20 0.46
AURKA O14965 1/20 0.46
DCLK1 O15075 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7880244 0.95 BRAF (0.44) BRAFCYP2C9RIPK2RAF1KDR
SCHEMBL7872497 0.87 BRAF (0.56) BRAFCYP2C9RIPK2RAF1KDR
SCHEMBL7876453 0.84 BTK (0.42) NEK2STK16MAP2K4PAK1TNIK
SCHEMBL298639 0.84 BRAF (0.54) BRAFCYP2C9RIPK2RAF1KDR
SCHEMBL299283 0.84 BRAF (0.69) BRAFCYP2C9RIPK2RAF1KDR
SCHEMBL7869167 0.83 CYP2C9 (0.44) CYP2C9CLK1CYP2C19CYP3A4CYP2D6
SCHEMBL7874309 0.83 EGFR (0.44) BRAFCYP2C9KDRFGFR1CYP3A4
SCHEMBL7878749 0.83 BRAF (0.50) BRAFCYP2C9RIPK2RAF1KDR
SCHEMBL7868957 0.82 CYP3A4 (0.51) CYP2C9CYP2C19CYP3A4
SCHEMBL19565631 0.82 BRAF (0.61) BRAFCYP2C9RIPK2RAF1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010129570-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS PLEXXIKON, INC. (US) 2010-11-11 WO disclosed