SCHEMBL7869167

SCHEMBL7869167

CN/C=C(\C=N)c1cnc2[nH]cc(C(=O)c3cccc(NS(=O)(=O)c4ccc(F)cc4)c3)c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 5/20 0.44
CYP3A4 P08684 4/20 0.44
CYP2C19 P33261 4/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
CYP1A2 P05177 1/20 0.44
GAA P10253 1/20 0.44
CYP2D6 P10635 1/20 0.44
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 1/20 0.44
PIK3CA P42336 1/20 0.43
CLK1 P49759 1/20 0.42
DYRK1A Q13627 1/20 0.42
BTK Q06187 1/20 0.42
ITGA1 P56199 2/20 0.41
HSD17B1 P14061 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7868957 0.93 CYP3A4 (0.51) CYP2C9CYP3A4CYP2C19SMN1; SMN2LMNA
SCHEMBL7874309 0.92 EGFR (0.44) CYP2C9CYP3A4LMNAMEN1MAPT
SCHEMBL7875675 0.91 BRD4 (0.42) CYP2C9CYP3A4SMN1; SMN2LMNAMEN1
SCHEMBL7880231 0.84 CYP3A4 (0.53) CYP2C9CYP3A4CYP2C19SMN1; SMN2LMNA
SCHEMBL298104 0.83 CYP2C9 (0.53) CYP2C9CYP3A4CYP2C19SMN1; SMN2LMNA
SCHEMBL7869103 0.83 BRAF (0.49) CYP2C9CYP3A4CYP2C19CYP2D6CLK1
SCHEMBL7876453 0.83 BTK (0.42) PIK3CABTK
SCHEMBL7880244 0.82 BRAF (0.44) CYP2C9CYP3A4CYP2C19CYP2D6CLK1
SCHEMBL7869096 0.82 CYP3A4 (0.45) CYP2C9CYP3A4CYP2C19LMNAMEN1
SCHEMBL7869062 0.80 CYP3A4 (0.44) CYP2C9CYP3A4SMN1; SMN2LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010129570-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS PLEXXIKON, INC. (US) 2010-11-11 WO disclosed