SCHEMBL7869911

SCHEMBL7869911

Fc1ccc(C2CCN(C[C@@H]3CN(Cc4cccc5ccccc45)C[C@H]3c3ccsc3)CC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 10/20 0.52
OPRM1 P35372 2/20 0.43
OPRK1 P41145 2/20 0.43
OPRL1 P41146 2/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
ACHE P22303 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7869741 1.00 CCR5 (0.52) CCR5OPRM1OPRK1OPRL1MEN1
SCHEMBL7874871 0.93 CCR5 (0.60) CCR5MEN1KMT2AACHE
SCHEMBL7872050 0.87 CCR5 (0.54) CCR5OPRM1MEN1KMT2A
SCHEMBL7872048 0.87 CCR5 (0.54) CCR5OPRM1MEN1KMT2A
SCHEMBL7869852 0.86 CCR5 (0.52) CCR5
SCHEMBL7871412 0.86 CCR5 (0.50) CCR5
SCHEMBL7869851 0.86 CCR5 (0.52) CCR5
SCHEMBL7871415 0.86 CCR5 (0.50) CCR5
SCHEMBL7871883 0.85 SLC6A4 (0.42) CCR5SLC6A4SLC6A3
SCHEMBL7868460 0.85 CCR5 (0.67) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303593-B1 FOR THERAPY HUMAN IMMUNODEFICIENCY VIRUS INFECTION, AQUIRED IMMUNODEFICIENCY SYNDROME (AIDS), INFLAMMATORY AND IMMUNOREGULATORY DISORDER OR DISEASE, ASTHMA, ALLERGIC RHINITIS, DERMATITIS, CONJUNCTIVITIS, ATHEROSCLEROSIS MERCK & CO., INC. 2001-10-16 US claimed
US-6303593-B1 FOR THERAPY HUMAN IMMUNODEFICIENCY VIRUS INFECTION, AQUIRED IMMUNODEFICIENCY SYNDROME (AIDS), INFLAMMATORY AND IMMUNOREGULATORY DISORDER OR DISEASE, ASTHMA, ALLERGIC RHINITIS, DERMATITIS, CONJUNCTIVITIS, ATHEROSCLEROSIS MERCK & CO., INC. 2001-10-16 US disclosed