SCHEMBL7870085

SCHEMBL7870085

CCc1cnc(-c2ccc(C)nc2C(=O)N2C[C@@H]3C[C@@H]3CC2COc2ccc(C(F)(F)F)cn2)o1

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 13/20 0.48
HCRTR2 O43614 9/20 0.47
CYP3A4 P08684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL609341 1.00 HCRTR1 (0.48) HCRTR1HCRTR2CYP3A4
SCHEMBL608175 0.87 HCRTR1 (0.54) HCRTR1HCRTR2
SCHEMBL7913236 0.87 CYP3A4 (0.54) HCRTR1HCRTR2CYP3A4
SCHEMBL3390051 0.87 CYP3A4 (0.54) HCRTR1HCRTR2CYP3A4
SCHEMBL610803 0.85 HCRTR1 (0.50) HCRTR1HCRTR2
SCHEMBL610097 0.85 CYP3A4 (0.54) HCRTR1HCRTR2CYP3A4
SCHEMBL7869499 0.85 CYP3A4 (0.54) HCRTR1HCRTR2CYP3A4
SCHEMBL608587 0.85 HCRTR1 (0.65) HCRTR1HCRTR2
SCHEMBL10121671 0.83 HCRTR2 (0.64) HCRTR1HCRTR2
SCHEMBL611060 0.83 HCRTR2 (0.64) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010122151-A1 3 -AZABICYCLO [4.1.0] HEPTANES USED AS OREXIN ANTAGONISTS GLAXO GROUP LIMITED (GB) 2010-10-28 WO disclosed