SCHEMBL7871808

SCHEMBL7871808

Cn1c(-c2ccccc2)cnc1[C@H]1CNCC[C@H]1O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.45
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
HPGDS O60760 3/20 0.38
SLC18A3 Q16572 2/20 0.37
GAA P10253 2/20 0.36
LDLR P01130 1/20 0.36
PCSK9 Q8NBP7 1/20 0.36
LMNA P02545 1/20 0.36
ATP1A1 P05023 3/20 0.35
ATP1B1 P05026 3/20 0.35
ATP1A3 P13637 3/20 0.35
ATP1B2 P14415 3/20 0.35
ATP1A2 P50993 3/20 0.35
ATP1B3 P54709 3/20 0.35
FXYD2 P54710 3/20 0.35
ATP1A4 Q13733 3/20 0.35
PIM1 P11309 1/20 0.35
PIM3 Q86V86 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27217014 0.74 CYP1A2 (0.51) CYP1A2CYP3A4CYP2D6HPGDSGAA
SCHEMBL27217262 0.73 CYP1A2 (0.54) CYP1A2CYP3A4CYP2D6HPGDSGAA
SCHEMBL27217047 0.73 CYP1A2 (0.50) CYP1A2CYP3A4CYP2D6HPGDSGAA
SCHEMBL10964453 0.68 SLC18A3 (0.54) HTR2ASLC18A3
SCHEMBL5923778 0.68 SLC18A3 (0.54) HTR2ASLC18A3
SCHEMBL10964458 0.68 SLC18A3 (0.54) HTR2ASLC18A3
SCHEMBL8273744 0.68 SLC18A3 (0.54) HTR2ASLC18A3
SCHEMBL10964208 0.68 SLC18A3 (0.54) HTR2ASLC18A3
SCHEMBL27217188 0.68 CYP1A2 (0.47) CYP1A2CYP3A4CYP2D6HPGDSGAA
SCHEMBL27217268 0.65 CYP1A2 (0.47) CYP1A2CYP3A4CYP2D6HPGDSGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed