SCHEMBL7872020

SCHEMBL7872020

O=C(c1cccc2cccnc12)N1CC(CN2CCC(c3ccc(F)cc3)CC2)C(c2ccsc2)C1

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 19/20 0.53
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7871992 0.93 CCR5 (0.63) CCR5
SCHEMBL7868367 0.89 CCR5 (0.54) CCR5
SCHEMBL7863002 0.87 CCR5 (0.71) CCR5
SCHEMBL7863001 0.87 CCR5 (0.71) CCR5
SCHEMBL7871152 0.86 CCR5 (0.51) CCR5
SCHEMBL7868243 0.85 CCR5 (0.51) CCR5
SCHEMBL7868244 0.85 CCR5 (0.51) CCR5
SCHEMBL7863126 0.85 CCR5 (0.62) CCR5
SCHEMBL7871880 0.85 CCR5 (0.57) CCR5
SCHEMBL7863141 0.84 CCR5 (0.53) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303593-B1 FOR THERAPY HUMAN IMMUNODEFICIENCY VIRUS INFECTION, AQUIRED IMMUNODEFICIENCY SYNDROME (AIDS), INFLAMMATORY AND IMMUNOREGULATORY DISORDER OR DISEASE, ASTHMA, ALLERGIC RHINITIS, DERMATITIS, CONJUNCTIVITIS, ATHEROSCLEROSIS MERCK & CO., INC. 2001-10-16 US claimed
US-6303593-B1 FOR THERAPY HUMAN IMMUNODEFICIENCY VIRUS INFECTION, AQUIRED IMMUNODEFICIENCY SYNDROME (AIDS), INFLAMMATORY AND IMMUNOREGULATORY DISORDER OR DISEASE, ASTHMA, ALLERGIC RHINITIS, DERMATITIS, CONJUNCTIVITIS, ATHEROSCLEROSIS MERCK & CO., INC. 2001-10-16 US disclosed