SCHEMBL7872974

SCHEMBL7872974

COC(=O)Cn1cnc2c(NC(c3ccccc3)(c3ccccc3)c3ccc(OC)cc3)ncnc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.47
HDAC6 Q9UBN7 1/20 0.47
FLT4 P35916 1/20 0.47
KDR P35968 1/20 0.47
HPGD P15428 1/20 0.44
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
HDAC2 Q92769 3/20 0.40
EGFR P00533 1/20 0.40
KMT2A Q03164 2/20 0.39
NSD3 Q9BZ95 1/20 0.39
CCNB2 O95067 1/20 0.39
CDK1 P06493 1/20 0.39
CCNB1 P14635 1/20 0.39
CCNB3 Q8WWL7 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA2B P29275 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7872820 0.93 HDAC1 (0.48) HDAC1HDAC6FLT4KDRHPGD
SCHEMBL21317389 0.81 CDK1 (0.50) HDAC1HDAC6HPGDCCNB2CDK1
SCHEMBL9230643 0.81 HDAC6 (0.58) HDAC1HDAC6FLT4KDRNSD3
SCHEMBL7867774 0.80 HSP90AA1 (0.39) HDAC1FLT4KDRHDAC2KMT2A
SCHEMBL7878997 0.77 DOT1L (0.35) HDAC1HDAC6FLT4KDRHPGD
SCHEMBL14175360 0.77 CDK1 (0.48) PDE4DTDP1EGFRCCNB2CDK1
SCHEMBL14175378 0.77 CCNB2 (0.46) HDAC1HDAC6HPGDEGFRCCNB2
SCHEMBL7166671 0.77 NSD3 (0.43) HDAC1HDAC6HPGDPDE4APDE4B
SCHEMBL8150599 0.77 HDAC1 (0.35) HDAC1HDAC6FLT4KDRHPGD
SCHEMBL9583386 0.75 CDK1 (0.44) HDAC1HDAC6KMT2ACCNB2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316595-B1 PNA synthesis using a base-labile amino protecting group AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-11-13 US disclosed
US-6121418-A PNA synthesis using a base-labile amino protecting group HOECHST AKTIENGESELLSCHAFT (DE) 2000-09-19 US disclosed