SCHEMBL9230643

SCHEMBL9230643

COC(=O)Cn1cnc2c(NC(=O)c3ccc(OC)cc3)ncnc21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.58
HDAC1 Q13547 1/20 0.58
BRD4 O60885 1/20 0.48
FLT4 P35916 1/20 0.46
KDR P35968 1/20 0.46
CDK5 Q00535 2/20 0.46
CDK5R1 Q15078 2/20 0.46
F2 P00734 1/20 0.44
F10 P00742 1/20 0.43
DEGS1 O15121 1/20 0.43
NSD3 Q9BZ95 1/20 0.42
NPC1 O15118 2/20 0.42
TP53 P04637 1/20 0.42
ALOX15 P16050 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CCNB2 O95067 1/20 0.42
CDK1 P06493 1/20 0.42
CCNB1 P14635 1/20 0.42
CCNB3 Q8WWL7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6748343 0.91 HDAC1 (0.58) HDAC6HDAC1BRD4FLT4KDR
SCHEMBL21011277 0.83 BRD4 (0.56) HDAC6HDAC1BRD4CDK5CDK5R1
SCHEMBL7872974 0.81 HDAC1 (0.47) HDAC6HDAC1FLT4KDRNSD3
SCHEMBL8646398 0.80 FLT4 (0.50) HDAC1FLT4KDRRAB9AALDH1A1
SCHEMBL26230949 0.79 FLT4 (0.49) HDAC6HDAC1FLT4KDRTMIGD3
SCHEMBL14192925 0.78 HDAC1 (0.48) HDAC6HDAC1TMIGD3
SCHEMBL3254930 0.77 RET (0.55) BRD4KDRF2DEGS1NPC1
SCHEMBL3457849 0.77 EGFR (0.54) HDAC1BRD4FLT4KDRNPC1
SCHEMBL6046940 0.76 HDAC1 (0.43) HDAC6HDAC1BRD4FLT4KDR
SCHEMBL14192930 0.76 HDAC6 (0.47) HDAC6HDAC1FLT4KDRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0672661-A1 Substituted N-ethyl-glycinderivatives for the preparation of PNA and PNA-/DNA hybrides HOECHST AKTIENGESELLSCHAFT (DE) 1995-09-20 EP disclosed