SCHEMBL787325

SCHEMBL787325

CC(C(=O)OC(=O)CCc1ccccc1)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.57
FFAR1 O14842 1/20 0.48
ALDH1A1 P00352 1/20 0.47
KEAP1 Q14145 1/20 0.46
KMT2A Q03164 2/20 0.46
RECQL P46063 1/20 0.45
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.44
MEN1 O00255 1/20 0.44
TRPV1 Q8NER1 1/20 0.44
ALOX5 P09917 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16440023 0.85 TDP1 (0.62) TDP1FFAR1ALDH1A1KEAP1KMT2A
Methyl 3-Phenylpropanoate SCHEMBL28962931 0.85 TDP1 (0.54) TDP1FFAR1ALDH1A1KMT2ARECQL
SCHEMBL28532192 0.84 ALDH1A1 (0.45) ALDH1A1KMT2ARECQLMAPTRAB9A
SCHEMBL5692495 0.82 CYP1A2 (0.45) ALDH1A1KMT2AMEN1
SCHEMBL28004226 0.80 TDP1 (0.56) TDP1FFAR1ALDH1A1KEAP1KMT2A
SCHEMBL1739439 0.79 TDP1 (0.73) TDP1FFAR1ALDH1A1KEAP1KMT2A
SCHEMBL5692490 0.79 KMT2A (0.52) KMT2A
SCHEMBL19094376 0.79 HCAR2 (0.50) TDP1ALDH1A1RAB9A
SCHEMBL8066953 0.79 HCAR2 (0.50) TDP1ALDH1A1RAB9A
SCHEMBL9074425 0.78 ALDH1A1 (0.55) TDP1FFAR1ALDH1A1KEAP1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616069-A1 ESTER PRO-DRUGS OF [3-(1-(1H-IMIDAZOL-4-YL)ETHYL)-2-METHYLPHENYL]METHANOL Allergan, Inc. (US) 2013-07-24 EP disclosed
EP-2616066-A1 ESTER PRO-DRUGS OF [3-(1-(1H-IMIDAZOL-4-YL)ETHYL)-2-METHYLPHENYL]METHANOL FOR TREATING RETINAL DISEASES Allergan, Inc. (US) 2013-07-24 EP disclosed
EP-2616067-A1 ESTER PRO-DRUGS OF [3-(1-(1H-IMIDAZOL-4-YL)ETHYL)-2-METHYLPHENYL]METHANOL FOR TREATING SKIN DISEASES AND CONDITIONS Allergan, Inc. (US) 2013-07-24 EP disclosed
WO-2012037484-A1 ESTER PRO-DRUGS OF [3-(1-(1H-IMIDAZOL-4-YL)ETHYL)-2-METHYLPHENYL] METHANOL FOR TREATING SKIN DISEASES AND CONDITIONS ALLERGAN, INC. (US) 2012-03-22 WO disclosed
WO-2012037453-A1 ESTER PRO-DRUGS OF [3-(1-(1H-IMIDAZOL-4-YL)ETHYL)-2-METHYLPHENYL] METHANOL FOR TREATING RETINAL DISEASES ALLERGAN, INC. (US) 2012-03-22 WO disclosed
WO-2012037499-A1 ESTER PRO-DRUGS OF [3-(1-(1H-IMIDAZOL-4-YL)ETHYL)-2-METHYLPHENYL] METHANOL ALLERGAN, INC. (US) 2012-03-22 WO disclosed