SCHEMBL7873423

SCHEMBL7873423

CC(Cc1ccc2c(c1)CCO2)C(C)NCC1CCN(C(=O)CCNS(C)(=O)=O)CC1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.46
MCHR1 Q99705 2/20 0.37
NPY5R Q15761 5/20 0.37
ACACB O00763 2/20 0.37
F2 P00734 1/20 0.35
PRSS1 P07477 1/20 0.35
PRSS2 P07478 1/20 0.35
PRSS3 P35030 1/20 0.35
S1PR1 P21453 1/20 0.35
FAAH O00519 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CHRM5 P08912 1/20 0.35
OGA O60502 1/20 0.35
HSD11B1 P28845 1/20 0.34
NPC1 O15118 1/20 0.34
POLB P06746 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4680284 0.88 CYP2D6 (0.43) CYP2D6MCHR1NPY5RACACBFAAH
SCHEMBL4681946 0.86 CYP2D6 (0.51) CYP2D6MCHR1ACACBCHRM5
SCHEMBL4682240 0.84 SIGMAR1 (0.40) CYP2D6MCHR1NPY5RACACBNPC1
SCHEMBL4678895 0.84 CYP2D6 (0.47) CYP2D6MCHR1ACACBFAAHCHRM5
Hydrochloric Acid SCHEMBL4684973 0.83 CYP2D6 (0.45) CYP2D6MCHR1NPY5RACACBF2
SCHEMBL4683509 0.83 CYP2D6 (0.51) CYP2D6MCHR1ACACBCHRM5OGA
SCHEMBL4679086 0.83 CYP2D6 (0.70) CYP2D6MCHR1ACACBF2PRSS1
SCHEMBL4679079 0.83 CYP2D6 (0.70) CYP2D6MCHR1ACACBF2PRSS1
SCHEMBL4680280 0.68 CYP2D6 (0.68) CYP2D6MCHR1ACACBFAAHSMN1; SMN2
SCHEMBL4680274 0.68 CYP2D6 (0.68) CYP2D6MCHR1ACACBFAAHSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6319920-B1 MUSCARINIC RECEPTOR ANTAGONIST USED IN GASTROINTESTINAL, GENITOURINARY TRACT, RESPIRATORY TRACT, CARDIOVASCULAR SYSTEM, CENTRAL NERVOUS SYSTEM DISORDERS AND IN ANESTHESIOLOGY AND OPHTHALMOLOGY SYNTEX (U.S.A.) LLC 2001-11-20 US claimed
US-6319920-B1 MUSCARINIC RECEPTOR ANTAGONIST USED IN GASTROINTESTINAL, GENITOURINARY TRACT, RESPIRATORY TRACT, CARDIOVASCULAR SYSTEM, CENTRAL NERVOUS SYSTEM DISORDERS AND IN ANESTHESIOLOGY AND OPHTHALMOLOGY SYNTEX (U.S.A.) LLC 2001-11-20 US disclosed