SCHEMBL7873587

SCHEMBL7873587

CC(N)Oc1cccc([N+](=O)[O-])c1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.52
LMNA P02545 2/20 0.52
CHRNB2 P17787 1/20 0.50
CHRNA4 P43681 1/20 0.50
ALDH1A1 P00352 2/20 0.49
ACHE P22303 1/20 0.49
F2 P00734 1/20 0.48
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
HGFAC Q04756 1/20 0.46
TP53 P04637 1/20 0.45
KMO O15229 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7671999 0.86 TSHR (0.55) TSHRLMNACHRNB2CHRNA4ALDH1A1
SCHEMBL27924572 0.83 TSHR (0.52) TSHRLMNACHRNB2CHRNA4ALDH1A1
SCHEMBL3879951 0.83 TSHR (0.52) TSHRLMNACHRNB2CHRNA4ALDH1A1
SCHEMBL20299326 0.83 TSHR (0.52) TSHRLMNACHRNB2CHRNA4ALDH1A1
SCHEMBL15994783 0.81 F2 (0.53) TSHRLMNACHRNB2CHRNA4ALDH1A1
SCHEMBL4998342 0.81 LMNA (0.54) TSHRLMNACHRNB2CHRNA4ALDH1A1
SCHEMBL11298055 0.81 MAPT (0.52) TSHRLMNACHRNB2CHRNA4ALDH1A1
SCHEMBL27771387 0.81 LMNA (0.54) TSHRLMNACHRNB2CHRNA4ALDH1A1
SCHEMBL27771390 0.81 TSHR (0.48) TSHRLMNACHRNB2CHRNA4ALDH1A1
SCHEMBL11248630 0.80 NPY5R (0.50) TSHRLMNACHRNB2CHRNA4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1067928-A4 METHODS FOR INHIBITING MRP1 LILLY CO ELI (US) 2001-11-14 EP disclosed
EP-1067928-A1 METHODS FOR INHIBITING MRP1 ELI LILLY AND COMPANY (US) 2001-01-17 EP disclosed
WO-1999051228-A1 METHODS FOR INHIBITING MRP1 ELI LILLY AND COMPANY (US) 1999-10-14 WO disclosed