SCHEMBL7874039

SCHEMBL7874039

C[C@@H](NC(=O)c1cc(C(=O)N[C@@H](Cc2ccccc2)[C@H](O)CNCC#CC2CC2)cc(N(C)[S+](C)[O-])c1)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 19/20 0.57
BACE2 Q9Y5Z0 6/20 0.57
CTSD P07339 2/20 0.57
APP P05067 1/20 0.57
CYP3A4 P08684 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8339052 0.79 BACE1 (0.58) BACE1BACE2CTSDAPP
SCHEMBL7880652 0.76 BACE1 (0.62) BACE1BACE2CTSDAPP
SCHEMBL7866943 0.76 BACE1 (0.50) BACE1BACE2CTSD
SCHEMBL8338864 0.73 BACE1 (0.46) BACE1BACE2CTSDAPP
SCHEMBL4216477 0.73 BACE1 (0.84) BACE1BACE2CTSDAPPCYP3A4
SCHEMBL20899826 0.73 BACE1 (1.00) BACE1BACE2CTSDAPP
SCHEMBL29470573 0.73 BACE1 (1.00) BACE1BACE2CTSDAPP
SCHEMBL21527047 0.73 BACE1 (1.00) BACE1BACE2CTSDAPP
SCHEMBL4567212 0.73 BACE1 (1.00) BACE1BACE2CTSDAPP
SCHEMBL8341359 0.73 BACE1 (0.45) BACE1BACE2CTSDAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010107384-A1 ASPARTYL PROTEASE INHIBITORS MEDIVIR AB (SE) 2010-09-23 WO disclosed