SCHEMBL7874849

SCHEMBL7874849

CN/C=C(\C=N)c1cnc2[nH]cc(C(=O)c3cc(NS(=O)(=O)C4CCCCC4)ccc3F)c2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 7/20 0.37
PAK1 Q13153 2/20 0.36
MAP2K4 P45985 2/20 0.36
BMPR1B O00238 1/20 0.36
PLK4 O00444 1/20 0.36
PIR O00625 1/20 0.36
AURKA O14965 1/20 0.36
DCLK1 O15075 1/20 0.36
EPHB6 O15197 1/20 0.36
RIPK2 O43353 1/20 0.36
STK16 O75716 1/20 0.36
OXSR1 O95747 1/20 0.36
MAP4K4 O95819 1/20 0.36
ABL1 P00519 1/20 0.36
RAF1 P04049 1/20 0.36
LCK P06239 1/20 0.36
FYN P06241 1/20 0.36
FES P07332 1/20 0.36
CSF1R P07333 1/20 0.36
YES1 P07947 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7876631 0.96 BRAF (0.38) BRAFPAK1MAP2K4BMPR1BPLK4
SCHEMBL298370 0.84 CYP2C19 (0.49) BRAFPAK1MAP2K4BMPR1BPLK4
SCHEMBL7876453 0.84 BTK (0.42) PAK1MAP2K4STK16NEK2TNIK
SCHEMBL298856 0.83 CYP2C19 (0.49) BRAFPAK1MAP2K4BMPR1BPLK4
SCHEMBL7872497 0.83 BRAF (0.56) BRAFPAK1MAP2K4BMPR1BPLK4
SCHEMBL7869096 0.82 CYP3A4 (0.45) BRAFPAK1MAP2K4BMPR1BPLK4
SCHEMBL7878749 0.82 BRAF (0.50) BRAFPAK1MAP2K4BMPR1BPLK4
SCHEMBL7880231 0.81 CYP3A4 (0.53) BRAFKITCYP2C19CYP2C9CYP3A4
SCHEMBL298381 0.79 BRAF (0.44) BRAFMAP2K4NEK2MAP2K1CYP2C9
SCHEMBL7869062 0.79 CYP3A4 (0.44) BRAFKITRIPK1CYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010129570-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS PLEXXIKON, INC. (US) 2010-11-11 WO disclosed