SCHEMBL7869062

SCHEMBL7869062

CN/C=C(\C=N)c1cnc2[nH]cc(C(=O)c3cc(NS(=O)(=O)c4cccc(C(F)(F)F)c4)ccc3F)c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.44
NTRK1 P04629 1/20 0.41
KIT P10721 1/20 0.41
HSD17B2 P37059 1/20 0.41
CYP2C9 P11712 2/20 0.40
MAPT P10636 4/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 2/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
TSHR P16473 1/20 0.38
GAA P10253 1/20 0.38
NR3C1 P04150 1/20 0.38
PGR P06401 1/20 0.38
AR P10275 1/20 0.38
ESR2 Q92731 1/20 0.38
PIK3CA P42336 1/20 0.38
RIPK1 Q13546 1/20 0.38
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7880231 0.91 CYP3A4 (0.53) CYP3A4KITCYP2C9HDAC1HDAC8
SCHEMBL7869096 0.90 CYP3A4 (0.45) CYP3A4KITHSD17B2CYP2C9MAPT
SCHEMBL7877658 0.89 CYP3A4 (0.42) CYP3A4KITCYP2C9HDAC1HDAC8
SCHEMBL298315 0.84 CYP3A4 (0.49) CYP3A4NTRK1KITHSD17B2CYP2C9
SCHEMBL7875675 0.84 BRD4 (0.42) CYP3A4NTRK1KITCYP2C9MAPT
SCHEMBL7868957 0.82 CYP3A4 (0.51) CYP3A4HSD17B2CYP2C9MAPTPOLB
SCHEMBL298650 0.81 BRAF (0.51) CYP3A4NTRK1KITHSD17B2MAPT
SCHEMBL7872497 0.81 BRAF (0.56) CYP3A4KITCYP2C9PGRRIPK1
SCHEMBL7876631 0.81 BRAF (0.38) CYP3A4KITCYP2C9RIPK1BRAF
SCHEMBL7869167 0.80 CYP2C9 (0.44) CYP3A4HSD17B2CYP2C9MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010129570-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS PLEXXIKON, INC. (US) 2010-11-11 WO disclosed