SCHEMBL7875415

SCHEMBL7875415

Oc1ccc2c(c1O)CC[C@@H]1NCC[C@H]21

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.61
HSD11B1 P28845 1/20 0.47
ADRA2A P08913 4/20 0.46
ADRA2B P18089 4/20 0.46
ADRA2C P18825 4/20 0.46
ADRA1D P25100 3/20 0.46
ADRA1A P35348 3/20 0.46
ADRA1B P35368 3/20 0.46
DRD1 P21728 1/20 0.44
DRD5 P21918 1/20 0.44
DRD3 P35462 1/20 0.44
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
ESR1 P03372 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
G6PD P11413 1/20 0.41
PKM P14618 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7874803 1.00 DRD2 (0.61) DRD2HSD11B1ADRA2AADRA2BADRA2C
SCHEMBL7886601 1.00 DRD2 (0.61) DRD2HSD11B1ADRA2AADRA2BADRA2C
SCHEMBL7880605 1.00 DRD2 (0.61) DRD2HSD11B1ADRA2AADRA2BADRA2C
Bromide SCHEMBL243103 0.98 DRD2 (0.60) DRD2HSD11B1ADRA2AADRA2BADRA2C
Bromide SCHEMBL240587 0.98 DRD2 (0.60) DRD2HSD11B1ADRA2AADRA2BADRA2C
Bromide SCHEMBL240352 0.98 DRD2 (0.60) DRD2HSD11B1ADRA2AADRA2BADRA2C
Bromide SCHEMBL239049 0.98 DRD2 (0.60) DRD2HSD11B1ADRA2AADRA2BADRA2C
SCHEMBL244216 0.90 DRD2 (0.76) DRD2HSD11B1ADRA2AADRA2BADRA2C
SCHEMBL241076 0.90 DRD2 (0.76) DRD2HSD11B1ADRA2AADRA2BADRA2C
SCHEMBL7885978 0.90 DRD2 (0.76) DRD2HSD11B1ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097087-A1 CATECHOLAMINE DERIVATIVES AND PRODRUGS THEREOF H. LUNDBECK A/S (DK) 2010-09-02 WO disclosed