SCHEMBL7876150

SCHEMBL7876150

CCc1ccc(C(CC(N)=O)NC(=O)c2ccccc2)cc1CC

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPT P10636 11/20 0.56
RXFP1 Q9HBX9 1/20 0.56
MAPK1 P28482 4/20 0.54
KMT2A Q03164 4/20 0.53
MEN1 O00255 3/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7876188 0.81 POLB (0.58) MAPTRXFP1MAPK1KMT2AMEN1
SCHEMBL7876133 0.81 NPSR1 (0.71) MAPTRXFP1MAPK1KMT2AMEN1
SCHEMBL7876448 0.71 POLB (0.58) MAPTKMT2AMEN1
SCHEMBL27553133 0.70 MEN1 (0.66) MAPTMAPK1KMT2AMEN1
SCHEMBL7867465 0.70 NPSR1 (0.57) MAPTRXFP1KMT2AMEN1
SCHEMBL7872611 0.70 NPSR1 (0.73) MAPTRXFP1KMT2AMEN1
SCHEMBL22995641 0.70 MEN1 (0.61) MAPTMAPK1KMT2AMEN1
SCHEMBL4659439 0.70 KDM4E (0.67) MAPK1KMT2AMEN1
SCHEMBL4660820 0.70 KDM4E (0.67) MAPK1KMT2AMEN1
SCHEMBL5642916 0.70 KDM4E (0.67) MAPK1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800505-B1 NOVEL IMMUNOTHERAPEUTIC ARYL AMIDES CELGENE CORP (US) 2001-09-26 EP claimed
US-5801195-A TUMOR NECROSIS AGENT INHIBITORS FOR COMBATING CACHEXIA, ENDOTOXIC SHOCK AND RETROVIRUS REPLICATION CELGENE CORPORATION (US) 1998-09-01 US claimed
US-5736570-A ADMINISTERING TO REDUCE TUMOR NECROSIS FACTOR (TNFA) LEVELS IN MAMMAL; RETROVIRAL DISEASE TREATMENT/PROPHYLAXIS CELGENE CORPORATION (US) 1998-04-07 US claimed
EP-0800505-B1 NOVEL IMMUNOTHERAPEUTIC ARYL AMIDES CELGENE CORP (US) 2001-09-26 EP disclosed
US-6046221-A USEFUL FOR REDUCING LEVELS OF TUMOR NECROSIS FACTOR-ALPHA IN A MAMMAL CELGENE CORPORATION (US) 2000-04-04 US disclosed
US-5801195-A TUMOR NECROSIS AGENT INHIBITORS FOR COMBATING CACHEXIA, ENDOTOXIC SHOCK AND RETROVIRUS REPLICATION CELGENE CORPORATION (US) 1998-09-01 US disclosed
US-5736570-A ADMINISTERING TO REDUCE TUMOR NECROSIS FACTOR (TNFA) LEVELS IN MAMMAL; RETROVIRAL DISEASE TREATMENT/PROPHYLAXIS CELGENE CORPORATION (US) 1998-04-07 US disclosed