SCHEMBL7876255

SCHEMBL7876255

CS(=O)(=O)c1ccc(-c2cnn(CC(F)(F)F)c(=O)c2NC2CCCO2)cc1

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 19/20 0.55
PTGS1 P23219 14/20 0.44
PLAT P00750 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4186541 0.86 PTGS2 (0.59) PTGS2PTGS1PLAT
SCHEMBL4180069 0.86 PTGS2 (0.59) PTGS2PTGS1PLAT
SCHEMBL4192320 0.86 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL4186485 0.85 PTGS2 (0.58) PTGS2PTGS1
SCHEMBL4189637 0.80 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL4187833 0.80 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL4177757 0.78 PTGS2 (0.57) PTGS2PTGS1PLAT
SCHEMBL4192319 0.78 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL4187837 0.77 PTGS2 (0.62) PTGS2PTGS1
SCHEMBL4192816 0.76 PTGS2 (0.70) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6307047-B1 PYRIDAZINONE COMPOUNDS; INHIBITORS OF CYCLOOXYGENASE-2 (COX-2); SELECTIVITY OF THESE COMPOUNDS FOR COX-2 MINIMIZES THE UNWANTED GI AND RENAL SIDE-EFFECTS SEEN WITH CURRENTLY MARKETED NON-STEROIDAL ANTI-INFLAMMATORY DRUGS ABBOTT LABORATORIES 2001-10-23 US disclosed