SCHEMBL7876450

SCHEMBL7876450

CS(=O)(=O)c1ccc(-c2c(-c3ccc(F)cc3)sc(C(=O)O)c2CO)cc1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 18/20 0.52
PTGS1 P23219 3/20 0.51
KDM4E B2RXH2 1/20 0.51
MT-CO1 P00395 1/20 0.51
MT-CO2 P00403 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
HPGD P15428 1/20 0.51
TSHR P16473 1/20 0.51
CYP2C19 P33261 1/20 0.51
HSD17B10 Q99714 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7874965 0.82 PTGS1 (0.45) PTGS2PTGS1
SCHEMBL6050740 0.81 PTGS2 (0.61) PTGS2PTGS1KDM4EMT-CO1MT-CO2
SCHEMBL6050737 0.79 PTGS2 (0.56) PTGS2PTGS1KDM4EMT-CO1MT-CO2
SCHEMBL9755841 0.77 PTGS2 (0.47) PTGS2PTGS1KDM4EMT-CO1MT-CO2
SCHEMBL7874913 0.77 PTGS2 (0.49) PTGS2PTGS1KDM4EMT-CO1MT-CO2
SCHEMBL6050867 0.76 PTGS2 (0.56) PTGS2PTGS1KDM4EMT-CO1MT-CO2
SCHEMBL6050692 0.76 PTGS2 (0.52) PTGS2PTGS1KDM4EMT-CO1MT-CO2
SCHEMBL6050686 0.76 PTGS2 (0.52) PTGS2PTGS1KDM4EMT-CO1MT-CO2
SCHEMBL6050619 0.75 PTGS2 (0.60) PTGS2PTGS1KDM4EHPGD
SCHEMBL6050699 0.75 PTGS2 (0.60) PTGS2PTGS1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329421-B1 PHENYL-SUBSTITUTED BENZOFURAN AND BENZOTHIOPHENE DERIVATIVES; NONSTEROIDAL ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA & CO. (CA) 2001-12-11 US disclosed
EP-0778834-B1 DIARYL BICYCLIC HETEROCYCLES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA INC (CA) 2000-01-26 EP disclosed
EP-0778834-A1 DIARYL BICYCLIC HETEROCYCLES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA INC. (CA) 1997-06-18 EP disclosed
US-5521213-A NONSTEROID ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA, INC. (CA) 1996-05-28 US disclosed
WO-1996006840-A1 DIARYL BICYCLIC HETEROCYCLES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA INC. (CA) 1996-03-07 WO disclosed