SCHEMBL7876707

SCHEMBL7876707

CS(=O)(=O)CCNc1cc(N2C3CCC2COC3)nc(-c2ccc(N=O)cc2)n1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ATR Q13535 2/20 0.37
MTOR P42345 13/20 0.35
PIK3CA P42336 11/20 0.35
PIK3CG P48736 1/20 0.34
PTGS2 P35354 4/20 0.33
BRD4 O60885 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL629451 0.90 PTGS2 (0.39) ATRMTORPIK3CAPIK3CGPTGS2
SCHEMBL629371 0.85 MEN1 (0.43) ATRMTORPIK3CAPIK3CGPTGS2
SCHEMBL627851 0.82 MTOR (0.53) MTORPIK3CAPIK3CG
SCHEMBL628413 0.79 PIK3CA (0.56) MTORPIK3CAPIK3CG
SCHEMBL7883148 0.79 CYP1A2 (0.49) PTGS2
SCHEMBL628562 0.78 PIK3CA (0.64) MTORPIK3CAPIK3CG
SCHEMBL628601 0.77 PIK3CA (0.66) MTORPIK3CAPIK3CG
SCHEMBL629216 0.76 MTOR (0.67) MTORPIK3CAPIK3CG
SCHEMBL9607534 0.76 MTOR (0.38) ATRMTORPIK3CAPIK3CG
SCHEMBL628448 0.69 PIK3CA (0.42) ATRMTORPIK3CAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010120998-A1 PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH LLC (US) 2010-10-21 WO disclosed