SCHEMBL7877599

SCHEMBL7877599

CN/C=C(\C=N)c1cnc2[nH]cc(C(=O)c3cccc(N)c3)c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 1/20 0.42
NEK2 P51955 3/20 0.40
BRD4 O60885 2/20 0.39
GSK3B P49841 2/20 0.39
NPC1 O15118 1/20 0.38
MITF O75030 1/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
PAK1 Q13153 2/20 0.38
AXL P30530 5/20 0.38
KDR P35968 3/20 0.38
NTRK1 P04629 3/20 0.38
DYRK1A Q13627 2/20 0.38
CDC7 O00311 1/20 0.38
PLK4 O00444 1/20 0.38
CHEK1 O14757 1/20 0.38
AURKA O14965 1/20 0.38
MAPK13 O15264 1/20 0.38
PDPK1 O15530 1/20 0.38
DYRK3 O43781 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7875473 0.85 BRAF (0.41) AAK1NEK2BRD4PAK1KDR
SCHEMBL3705033 0.81 AAK1 (0.47) AAK1NEK2BRD4GSK3BNPC1
SCHEMBL297839 0.81 AAK1 (0.45) AAK1NEK2BRD4GSK3BNPC1
SCHEMBL7869103 0.80 BRAF (0.49) NEK2PAK1KDRPLK4AURKA
SCHEMBL7876453 0.80 BTK (0.42) AAK1NEK2BRD4GSK3BPAK1
SCHEMBL298022 0.79 PAK1 (0.48) AAK1NEK2BRD4GSK3BNPC1
SCHEMBL297306 0.79 BRAF (0.45) AAK1NEK2BRD4GSK3BNPC1
SCHEMBL3698741 0.78 AAK1 (0.53) AAK1NEK2BRD4GSK3BNPC1
SCHEMBL7880244 0.78 BRAF (0.44) NEK2PAK1KDRPLK4AURKA
SCHEMBL7874309 0.78 EGFR (0.44) LMNAKDREGFRFGFR1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010129570-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS PLEXXIKON, INC. (US) 2010-11-11 WO disclosed