SCHEMBL7877972

SCHEMBL7877972

CCCCCC(C)(C#N)CO

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.35
FDPS P14324 11/20 0.33
GGPS1 O95749 7/20 0.33
LMNA P02545 2/20 0.33
TSHR P16473 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CES2 O00748 1/20 0.31
LPAR1 Q92633 1/20 0.31
LPAR3 Q9UBY5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9183342 0.93 TSHR (0.33) SMN1; SMN2FDPSTSHRALDH1A1
SCHEMBL366645 0.86 TSHR (0.38) FDPSGGPS1TSHRCES2LPAR1
SCHEMBL28930082 0.84 TSHR (0.40) FDPSGGPS1TSHRCES2LPAR1
SCHEMBL28191748 0.84 TSHR (0.40) FDPSGGPS1TSHRCES2LPAR1
SCHEMBL10029661 0.84 TSHR (0.40) FDPSGGPS1TSHRCES2LPAR1
SCHEMBL9912385 0.84 TSHR (0.40) FDPSGGPS1TSHRCES2LPAR1
SCHEMBL20967951 0.84 TSHR (0.40) FDPSGGPS1TSHRCES2LPAR1
SCHEMBL12208739 0.84 TSHR (0.40) FDPSGGPS1TSHRCES2LPAR1
SCHEMBL9186812 0.84
Boric Acid SCHEMBL27917318 0.83 FDPS (0.33) FDPSGGPS1TSHRCES2LPAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174888-B1 POTENT PURINE NUCLEOSIDE PHOSPHORYLASE INHIBITORS; INHIBITORS OF T-CELL FORMATION, I.E., IMMUNOSUPPRESSANTS; TRANSPLANT REJECTION; AUTOIMMUNE DISEASES, E.G., RHEUMATOID DISEASES, PSORIASIS, DERMATITIS, CROHN'S DISEASE, UVEITIS; NOVARTIS AG (CH) 2001-01-16 US disclosed
US-6043365-A REACTING BIARYL OR CARBOCYCLIC OR HETEROCYCLIC ISOPROPYL NITRILE DERIVATIVE WITH A LOWER ALKYL ESTER OF FORMIC ACID, CONDENSING THE INTERMEDIATE FORMED WITH AN AMINOALKYL ESTER TO OBTAIN INTERMEDIATE, CYCLIZING AND CONDENSING NOVARTIS AG (CH) 2000-03-28 US disclosed
EP-0986563-A1 2-AMINO-7-(1-SUBSTITUTED-2-HYDROXYETHYL)-3,5-DIHYDRO-PYRROLO 3,2-D]PYRIMIDIN-4-ONES Novartis AG (CH) 2000-03-22 EP disclosed
WO-1998054185-A1 2-AMINO-7-(1-SUBSTITUTED-2-HYDROXYETHYL)-3,5-DIHYDRO-PYRROLO[3,2-D]PYRIMIDIN-4-ONES NOVARTIS AG (CH) 1998-12-03 WO disclosed