SCHEMBL78784

SCHEMBL78784

CC[C@@H]1C(C(=O)N(Cc2cccc(Cl)c2Cl)C2CC2)=C(c2ccc(OCCOc3c(F)ccc(F)c3Cl)cc2)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.61

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
REN P00797 19/20 0.61
CYP3A4 P08684 3/20 0.53
CTSD P07339 1/20 0.51
CTSE P14091 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL78486 0.94 CYP3A4 (0.54) RENCYP3A4
SCHEMBL78462 0.92 CYP3A4 (0.52) RENCYP3A4
SCHEMBL66311 0.91 REN (0.59) RENCYP3A4CTSDCTSE
SCHEMBL66312 0.91 REN (0.59) RENCYP3A4CTSDCTSE
SCHEMBL78833 0.91 CYP3A4 (0.61) RENCYP3A4
SCHEMBL65821 0.89 CYP3A4 (0.54) RENCYP3A4
SCHEMBL65820 0.89 CYP3A4 (0.54) RENCYP3A4
SCHEMBL65228 0.88 CYP3A4 (0.53) RENCYP3A4
SCHEMBL65227 0.88 CYP3A4 (0.53) RENCYP3A4
SCHEMBL79513 0.88 REN (0.46) RENCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed