SCHEMBL7878403

SCHEMBL7878403

COCc1nc(C(C)(C)O)c(C(=O)O)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 6/20 0.58
AGTR2 P50052 5/20 0.58
ABCC3 O15438 1/20 0.47
ABCC4 O15439 1/20 0.47
ABCB11 O95342 1/20 0.47
CYP3A4 P08684 1/20 0.47
PDE4D Q08499 1/20 0.47
PDE3A Q14432 1/20 0.47
SLCO1B3 Q9NPD5 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
SLCO1B1 Q9Y6L6 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7883521 0.92 AGTR1 (0.49) AGTR1AGTR2ABCC3ABCC4ABCB11
SCHEMBL7878593 0.92 AGTR1 (0.59) AGTR1AGTR2ABCC3ABCC4ABCB11
SCHEMBL7889758 0.91 AGTR1 (0.61) AGTR1AGTR2ABCC3ABCC4ABCB11
SCHEMBL7886561 0.91 AGTR1 (0.56) AGTR1AGTR2ABCC3ABCC4ABCB11
SCHEMBL7309878 0.91 AGTR1 (0.63) AGTR1AGTR2ABCC3ABCC4ABCB11
SCHEMBL7886530 0.90 AGTR1 (0.59) AGTR1AGTR2ABCC3ABCC4ABCB11
Olmesartan SCHEMBL94037 0.89 AGTR1 (0.73) AGTR1AGTR2ABCC3ABCC4ABCB11
Olmesartan SCHEMBL29368106 0.89 AGTR1 (0.73) AGTR1AGTR2ABCC3ABCC4ABCB11
Olmesartan SCHEMBL4221669 0.88 AGTR1 (0.72) AGTR1AGTR2ABCC3ABCC4ABCB11
SCHEMBL7889500 0.88 AGTR1 (0.58) AGTR1AGTR2ABCC3ABCC4ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0573218-B1 4-Carboxyimidazoles as angiotensin II antagonists and their thrapeutic use SANKYO CO (JP) 2001-03-07 EP claimed
CN-1051766-C Angiotensin II antagonist imidazole derivatives, their preparation and their theapeutic use SANKYO CO (JP) 2000-04-26 CN claimed
US-5646171-A HYPOTENSIVE AGENTS SANKYO COMPANY, LIMITED (JP) 1997-07-08 US claimed
EP-0573218-A2 4-Carboxyimidazoles as angiotensin II antagonists and their thrapeutic use SANKYO COMPANY LIMITED (JP) 1993-12-08 EP claimed
EP-0573218-B1 4-Carboxyimidazoles as angiotensin II antagonists and their thrapeutic use SANKYO CO (JP) 2001-03-07 EP disclosed
CN-1051766-C Angiotensin II antagonist imidazole derivatives, their preparation and their theapeutic use SANKYO CO (JP) 2000-04-26 CN disclosed
US-5646171-A HYPOTENSIVE AGENTS SANKYO COMPANY, LIMITED (JP) 1997-07-08 US disclosed
US-5616599-A HYPOTENSIVE AGENTS FOR CARDIOVASCULAR DISORDER SANKYO COMPANY, LIMITED (JP) 1997-04-01 US disclosed
EP-0573218-A2 4-Carboxyimidazoles as angiotensin II antagonists and their thrapeutic use SANKYO COMPANY LIMITED (JP) 1993-12-08 EP disclosed