SCHEMBL787889

SCHEMBL787889

CCCc1ccc2sc(S(=O)(=O)Nc3cccc(C(=O)OC)c3)c(C)c2c1

nearest known ligand 0.72

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PFKFB3 Q16875 14/20 0.72
PFKFB4 Q16877 12/20 0.72
CMA1 P23946 5/20 0.57
TCF4 P15884 1/20 0.50
CTNNB1 P35222 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL787986 0.84 PFKFB3 (1.00) PFKFB3PFKFB4CMA1TCF4CTNNB1
SCHEMBL787869 0.84 PFKFB3 (1.00) PFKFB3PFKFB4CMA1
SCHEMBL788203 0.84 PFKFB3 (0.77) PFKFB3PFKFB4CMA1TCF4CTNNB1
SCHEMBL787888 0.82 PFKFB3 (1.00) PFKFB3PFKFB4CMA1
SCHEMBL788389 0.80 PFKFB3 (0.56) PFKFB3PFKFB4TCF4CTNNB1
SCHEMBL788429 0.79 PFKFB3 (0.87) PFKFB3PFKFB4CMA1
SCHEMBL788154 0.79 PFKFB3 (0.83) PFKFB3PFKFB4CMA1
SCHEMBL787883 0.79 PFKFB3 (0.69) PFKFB3PFKFB4CMA1
SCHEMBL788058 0.79 PFKFB3 (1.00) PFKFB3PFKFB4CMA1
SCHEMBL806139 0.78 PFKFB3 (0.84) PFKFB3PFKFB4CMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616450-A2 SULFONAMIDE COMPOUNDS Kancera AB (SE) 2013-07-24 EP claimed
WO-2012035171-A2 NEW COMPOUNDS KANCERA AB (SE) 2012-03-22 WO claimed
WO-2020080979-A1 PFKFB3 INHIBITORS AND THEIR USES GERO DISCOVERY LIMITED LIABILITY COMPANY (RU) 2020-04-23 WO disclosed