SCHEMBL7879356

SCHEMBL7879356

COC(CCc1ccc(Br)cc1)c1nc(-c2ccccc2)oc1C

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.40
PPARG P37231 15/20 0.40
PPARA Q07869 12/20 0.40
TARBP2 Q15633 1/20 0.39
KDM4E B2RXH2 1/20 0.37
PPARD Q03181 2/20 0.37
RAB9A P51151 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7879351 1.00 FFAR1 (0.40) FFAR1PPARGPPARATARBP2KDM4E
SCHEMBL9436318 0.83 PPARG (0.43) FFAR1PPARGPPARATARBP2KDM4E
SCHEMBL7879344 0.70 PPARG (0.46) PPARGPPARATARBP2KDM4EPPARD
SCHEMBL7877729 0.70 PPARG (0.46) PPARGPPARATARBP2KDM4EPPARD
SCHEMBL4929594 0.70 KDM4E (0.47) PPARGPPARATARBP2KDM4ERAB9A
SCHEMBL9008061 0.69 KDM4E (0.41) PPARGPPARATARBP2KDM4EPPARD
SCHEMBL4918327 0.68 TARBP2 (0.46) PPARGPPARATARBP2KDM4ERAB9A
SCHEMBL7737637 0.68 KDM4E (0.46) PPARGPPARATARBP2KDM4ERAB9A
SCHEMBL17540833 0.68 KDM4E (0.49) PPARGPPARATARBP2KDM4ERAB9A
SCHEMBL4263081 0.67 NR1H4 (0.51) TARBP2KDM4ERAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329408-B1 HYPOCHOLESTEROLEMIC AGENTS; OPTICALLY PURE PFIZER INC. 2001-12-11 US disclosed
EP-0641338-A1 HYPOGLYCEMIC THIAZOLIDINEDIONES AND INTERMEDIATES PFIZER INC. (US) 1995-03-08 EP disclosed
WO-1993002079-A1 HYPOGLYCEMIC THIAZOLIDINEDIONES AND INTERMEDIATES PFIZER INC. (US) 1993-02-04 WO disclosed