SCHEMBL7879683

SCHEMBL7879683

CN(C(=N)N)C(=O)c1cc2ccc(Cl)cc2[nH]1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 7/20 0.55
HRH4 Q9H3N8 3/20 0.48
PDGFRB P09619 1/20 0.47
FLT3 P36888 1/20 0.47
PLG P00747 1/20 0.44
PLAU P00749 1/20 0.44
HAO1 Q9UJM8 1/20 0.43
F7 P08709 1/20 0.42
F3 P13726 1/20 0.42
DAO P14920 1/20 0.42
HRH3 Q9Y5N1 1/20 0.41
GPR183 P32249 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7884850 0.99 ALOX15 (0.53) ALOX15HRH4PDGFRBFLT3PLG
SCHEMBL7877877 0.89 HRH4 (0.61) HRH4FLT3F7F3HRH3
Hydrochloric Acid SCHEMBL7873360 0.88 HRH4 (0.60) HRH4FLT3F7F3HRH3
SCHEMBL7882071 0.85 FLT3 (0.49) PDGFRBFLT3PLGPLAUDAO
SCHEMBL7873326 0.85 HRH4 (0.47) HRH4PDGFRBFLT3PLGPLAU
SCHEMBL7873682 0.85 HRH4 (0.49) ALOX15HRH4PLGPLAU
Hydrochloric Acid SCHEMBL7882161 0.84 HRH4 (0.48) ALOX15HRH4PLGPLAU
Hydrochloric Acid SCHEMBL7880745 0.84 FLT3 (0.48) PDGFRBFLT3PLGPLAUDAO
Hydrochloric Acid SCHEMBL7881992 0.84 HRH4 (0.46) HRH4PDGFRBFLT3PLGPLAU
SCHEMBL7881464 0.82 FLT3 (0.54) HRH4PDGFRBFLT3DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248772-B1 HYPOTENSIVE AGENTS; ANTIARRHYTHMIA AGENTS; ANTIDIABETIC AGENTS; ANTIPROLIFERATIVE AGENTS SUMITOMO PHARMACEUTICALS CO., LTD. (JP) 2001-06-19 US disclosed
US-6169107-B1 USEFUL FOR THE TREATMENT AND PREVENTION OF DISEASES CAUSED BY INCREASED SODIUM/PROTON (NA.SUP.+ /H.SUP.+) EXCHANGER ACTIVITY, FOR EXAMPLE, HYPERTENSION, ARRHYTHMIA, ANGINA PECTORIS, CARDIAC HYPERTROPHY, DIABETES MELLITUS SUMITOMO PHARMACEUTICAL CO., LTD. (JP) 2001-01-02 US disclosed
EP-0622356-B1 Indoloylguanidine derivatives as inhibitors of sodium-hydrogen exchange SUMITOMO PHARMA (JP) 1998-07-01 EP disclosed
EP-0708091-A2 Indoloylguanidine derivatives SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1996-04-24 EP disclosed
EP-0622356-A1 Indoloylguanidine derivatives as inhibitors of sodium-hydrogen exchange SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1994-11-02 EP disclosed