SCHEMBL78797

SCHEMBL78797

CC[C@@H]1C(C(=O)N(Cc2cccc(Cl)c2Cl)C2CC2)C(=O)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
REN P00797 11/20 0.52
SLC6A4 P31645 5/20 0.43
KCNH2 Q12809 4/20 0.42
SLC6A2 P23975 4/20 0.41
CYP3A4 P08684 3/20 0.40
SLC6A3 Q01959 2/20 0.40
CYP2D6 P10635 1/20 0.40
GHSR Q92847 1/20 0.36
TSHR P16473 1/20 0.36
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65431 0.90 REN (0.49) RENSLC6A4KCNH2SLC6A2CYP3A4
SCHEMBL65432 0.90 REN (0.49) RENSLC6A4KCNH2SLC6A2CYP3A4
SCHEMBL3111265 0.80 REN (0.52) RENSLC6A4KCNH2SLC6A2CYP3A4
SCHEMBL78425 0.75 REN (0.43) RENCYP3A4
SCHEMBL78744 0.74 REN (0.43) RENSLC6A4CYP3A4
SCHEMBL78437 0.74 REN (0.42) RENSLC6A4CYP3A4
SCHEMBL79513 0.74 REN (0.46) RENCYP3A4
SCHEMBL78486 0.71 CYP3A4 (0.54) RENCYP3A4
SCHEMBL38659661 0.71 HSD17B10 (0.37)
SCHEMBL10182098 0.70 REN (0.49) RENSLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed