SCHEMBL7879807

SCHEMBL7879807

OC1CN(Cc2cccc(-c3ccccc3)c2)CCc2cc(OCc3ccccc3)ccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 16/20 1.00
GRIN2B Q13224 16/20 1.00
SIGMAR1 Q99720 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18587450 0.90 GRIN1 (0.81) GRIN1GRIN2BSIGMAR1
SCHEMBL3393477 0.81 GRIN2B (1.00) GRIN1GRIN2BSIGMAR1
SCHEMBL3392267 0.81 GRIN2B (1.00) GRIN1GRIN2BSIGMAR1
SCHEMBL3394898 0.78 GRIN1 (1.00) GRIN1GRIN2BSIGMAR1
SCHEMBL3396633 0.77 GRIN1 (1.00) GRIN1GRIN2BSIGMAR1
SCHEMBL3394795 0.77 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL3965085 0.76 GRIN1 (0.61) GRIN1GRIN2B
SCHEMBL3970687 0.76 GRIN1 (0.61) GRIN1GRIN2B
SCHEMBL1746466 0.76 GRIN1 (0.61) GRIN1GRIN2B
SCHEMBL3772950 0.74 GRIN1 (1.00) GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246331-A1 NR2B-selective NMDA-receptor antagonists Westfälische Wilhelms-Universität Münster (DE) 2010-11-03 EP disclosed
WO-2010122134-A1 NR2B-SELECTIVE NMDA-RECEPTOR ANTAGONISTS Westfälische Wilhelms Universität Münster (DE) 2010-10-28 WO disclosed