SCHEMBL788040

SCHEMBL788040

CS(=O)(=O)Cl.CS(=O)(=O)Oc1ccc2c(c1)CCC1C2CCC2C(=O)CCC21

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
STS P08842 13/20 0.47
ABCC4 O15439 3/20 0.47
ABCC1 P33527 2/20 0.47
KDM4E B2RXH2 2/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
CA9 Q16790 2/20 0.47
CYP2C9 P11712 1/20 0.47
SLCO1B1 Q9Y6L6 1/20 0.47
ESR1 P03372 1/20 0.47
CA4 P22748 1/20 0.47
CA6 P23280 1/20 0.47
ESR2 Q92731 1/20 0.47
CYP3A4 P08684 1/20 0.44
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
HSD17B1 P14061 1/20 0.43
RECQL P46063 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12826524 0.84 STS (0.61) STSCA1CA2CA9ESR1
SCHEMBL6569001 0.82 LMNA (0.60) STSABCC4ABCC1KDM4ECA1
SCHEMBL25529639 0.82 LMNA (0.60) STSABCC4ABCC1KDM4ECA1
SCHEMBL5499832 0.80 KDM4E (0.43) STSABCC4ABCC1KDM4ECA1
SCHEMBL5496755 0.79 STS (0.40) STSABCC4ABCC1KDM4ECA1
SCHEMBL22448486 0.78 LMNA (0.59) STSABCC4ABCC1KDM4ECA1
SCHEMBL773508 0.77 ESR1 (0.46) STSABCC4ABCC1KDM4ECA1
SCHEMBL773507 0.77 ESR1 (0.46) STSABCC4ABCC1KDM4ECA1
SCHEMBL17531381 0.74 STS (0.82) STSABCC4ABCC1KDM4ECA1
SCHEMBL8034430 0.74 STS (0.82) STSABCC4ABCC1KDM4ECA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616477-A2 6-SUBSTITUTED DEMETHYL-ESTRADIOL DERIVATIVES AS ER-BETA AGONISTS Endece, LLC (US) 2013-07-24 EP disclosed
WO-2012037261-A2 6-SUBSTITUTED DEMETHYL-ESTRADIOL DERIVATIVES AS ER-BETA AGONISTS ENDECE, LLC (US) 2012-03-22 WO disclosed