Camptothecin

Camptothecin

SCHEMBL788063

CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1.CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 18/20 1.00
ALDH1A1 P00352 4/20 1.00
MEN1 O00255 4/20 1.00
KMT2A Q03164 4/20 1.00
SMN1; SMN2 Q16637 4/20 1.00
KDM4E B2RXH2 3/20 1.00
GLA P06280 3/20 1.00
TP53 P04637 2/20 1.00
HPGD P15428 2/20 1.00
CYP3A4 P08684 2/20 1.00
HBB P68871 2/20 1.00
STAT6 P42226 1/20 1.00
CHEK1 O14757 1/20 1.00
HDAC3 O15379 1/20 1.00
ABCC4 O15439 1/20 1.00
GMNN O75496 1/20 1.00
LMNA P02545 1/20 1.00
CYP1A2 P05177 1/20 1.00
HNRNPA1 P09651 1/20 1.00
GAA P10253 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Camptothecin SCHEMBL29360250 1.00 TOP1 (1.00) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL29351099 1.00 TOP1 (1.00) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL28057307 1.00 TOP1 (1.00) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL29369924 1.00 TOP1 (1.00) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL4304557 1.00 TOP1 (1.00) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL6038 1.00 TOP1 (1.00) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL2298909 1.00 TOP1 (1.00) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL548833 0.99 TOP1 (0.98) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL17112859 0.99 TOP1 (0.98) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL3117386 0.99 TOP1 (0.98) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2854818-A2 CHEMICAL SUPPRESSORS OF NEUROTOXICITY IN SYNUCLEINOPATHIC DISEASES Oxalys Pharmaceuticals (CA) 2015-04-08 EP disclosed
WO-2013179144-A2 CHEMICAL SUPPRESSORS OF NEUROTOXICITY IN SYNUCLEINOPATHIC DISEASES OXALYS PHARMACEUTICALS (CA) 2013-12-05 WO disclosed
EP-2616484-A2 SCREENING METHOD Universiteit Leiden (NL) 2013-07-24 EP disclosed
WO-2012035120-A2 SCREENING METHOD UNIVERSITEIT LEIDEN (NL) 2012-03-22 WO disclosed
WO-2008070858-A1 INHIBITING TRANSLATION OF ABRERRANT DNMT3B TRANSCRIPTS IN CANCER CELLS USING INHIBITORY NUCLEIC ACIDS UNIVERSITY OF CHICAGO (US) 2008-06-12 WO disclosed
WO-2005082422-A1 COMBINATION OF AD-P53 AND CHEMOTHERAPY FOR THE TREATMENT OF TUMOURS INTROGEN THERAPEUTICS, INC. (US) 2005-09-09 WO disclosed
US-20050170015-A1 Antiproliferative colchicine compositions and uses thereof CHEMGENEX PHARMACEUTICALS, INC. 2005-08-04 US disclosed
EP-1330242-A2 ANTIPROLIFERATIVE COLCHICINE COMPOSITIONS AND USES THEREOF Chemgenex Therapeutics Inc. (US) 2003-07-30 EP disclosed
WO-2002056872-A2 ANTIPROLIFERATIVE COLCHICINE COMPOSITIONS AND USES THEREOF CHEMGENEX THERAPEUTICS, INC. (US) 2002-07-25 WO disclosed
WO-1991016904-A1 METHOD FOR TREATING RETROVIRAL INFECTIONS IN MAMMALS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, U.S. DEPARTMENT OF COMMERCE (US) 1991-11-14 WO disclosed