SCHEMBL7880673

SCHEMBL7880673

COC(=O)c1ccc(-c2ccnc(C)c2-c2ccc(N)nc2)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MTOR P42345 18/20 0.52
CCNE1 P24864 2/20 0.52
CDK2 P24941 2/20 0.52
GSK3A P49840 1/20 0.47
PIK3CA P42336 2/20 0.42
NPC1 O15118 1/20 0.39
MAPT P10636 1/20 0.39
NFKB1 P19838 1/20 0.39
RAB9A P51151 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PDK2 Q15119 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7872340 0.88 MTOR (0.55) MTORCCNE1CDK2GSK3APIK3CA
SCHEMBL7875765 0.88 MTOR (0.56) MTORCCNE1CDK2PIK3CA
SCHEMBL7883941 0.87 MTOR (0.50) MTORCCNE1CDK2PIK3CA
SCHEMBL12773632 0.85 MTOR (0.71) MTORCCNE1CDK2GSK3APIK3CA
SCHEMBL12137706 0.84 MTOR (0.46) MTORCCNE1CDK2PIK3CANPC1
SCHEMBL694987 0.83 MTOR (0.77) MTORCCNE1CDK2GSK3APIK3CA
SCHEMBL6893242 0.83 PIK3CA (0.56) MTORPIK3CA
SCHEMBL7871050 0.82 MTOR (0.47) MTOR
SCHEMBL12773417 0.81 MTOR (0.73) MTORCCNE1CDK2GSK3APIK3CA
SCHEMBL12773419 0.80 MTOR (0.73) MTORCCNE1CDK2GSK3APIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010122069-A1 5-ALKYNYL-PYRIDINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-10-28 WO disclosed