SCHEMBL7885461

SCHEMBL7885461

Clc1ccc2c(c1Cl)CCNCC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 13/20 1.00
HTR2C P28335 13/20 1.00
HTR2B P41595 12/20 1.00
PNMT P11086 6/20 0.75
ADRA2A P08913 1/20 0.75
ADRA2B P18089 1/20 0.75
ADRA2C P18825 1/20 0.75
NOTUM Q6P988 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30139643 0.86 HTR2A (0.75) HTR2AHTR2CHTR2BPNMTADRA2A
SCHEMBL6187756 0.86 HTR2A (0.75) HTR2AHTR2CHTR2BPNMTADRA2A
SCHEMBL1772370 0.86 PNMT (1.00) HTR2AHTR2CHTR2BPNMTADRA2A
Hydrochloric Acid SCHEMBL11211829 0.84 PNMT (1.00) HTR2AHTR2CHTR2BPNMTADRA2A
Hydrochloric Acid SCHEMBL11359434 0.84 PNMT (0.73) HTR2AHTR2CHTR2BPNMTADRA2A
SCHEMBL10227459 0.80 HTR2A (0.67) HTR2AHTR2CHTR2BPNMTADRA2A
SCHEMBL10228373 0.80 HTR2C (0.67) HTR2AHTR2CHTR2BPNMTADRA2A
SCHEMBL11947505 0.80 HTR2C (0.67) HTR2AHTR2CHTR2BPNMTADRA2A
SCHEMBL21762550 0.76 HTR2C (1.00) HTR2AHTR2CHTR2BPNMTADRA2A
SCHEMBL10879871 0.75 PNMT (0.75) HTR2AHTR2CHTR2BPNMTADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6172073-B1 BENZIMIDAZOLYLOXY ALKANAMINES AS SEROTONIN REUPTAKE INHIBITORS; NICOTINE AND TOBACCO WITHDRAWAL; PSYCHOLOGICAL, EATING, BRAIN, GASTROINTESTINAL, SLEEP, AND SEXUAL DISORDERS ELI LILLY AND COMPANY 2001-01-09 US disclosed
US-5789402-A Compounds having effects on serotonin-related systems ELI LILLY COMPANY (US) 1998-08-04 US disclosed
US-5741789-A HETERO-OXY ALKANAMINES ELI LILLY AND COMPANY (US) 1998-04-21 US disclosed
US-5627196-A ANTIDEPRESSANTS AND ANTISEROTONIN AGENTS ELI LILLY AND COMPANY (US) 1997-05-06 US disclosed
US-5614523-A INDOLYLOXY COMPOUNDS ELI LILLY AND COMPANY (US) 1997-03-25 US disclosed
US-5576321-A ALKOXY-SUBSTITUTED INDOLES ELI LILLY AND COMPANY (US) 1996-11-19 US disclosed
EP-0722941-A2 Compounds having effects on serotonin-related systems ELI LILLY AND COMPANY (US) 1996-07-24 EP disclosed