SCHEMBL7887017

SCHEMBL7887017

CCc1cc(C#N)ccc1/C=N/O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
CYP2A6 P11509 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
GAA P10253 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
PIN1 Q13526 1/20 0.38
SETDB1 Q15047 1/20 0.37
RAD51 Q06609 1/20 0.37
EGLN2 Q96KS0 1/20 0.36
PGR P06401 2/20 0.36
ABCC9 O60706 1/20 0.36
ABCC8 Q09428 1/20 0.36
KCNJ11 Q14654 1/20 0.36
KCNJ8 Q15842 1/20 0.36
TSHR P16473 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7887020 1.00 HPGD (0.40) HPGDALDH1A1MAPTCYP2A6KDM4E
SCHEMBL29952696 0.81 CYP2A6 (0.44) HPGDALDH1A1MAPTCYP2A6KDM4E
SCHEMBL1859259 0.81 CYP2A6 (0.44) HPGDALDH1A1MAPTCYP2A6KDM4E
SCHEMBL5045603 0.77 MAPT (0.46) HPGDALDH1A1MAPTKDM4EMEN1
SCHEMBL2463003 0.76 DYRK1A (0.38) HPGDALDH1A1MAPTCYP2A6KDM4E
SCHEMBL11306935 0.76 EGFR (0.41) ALDH1A1KDM4EMEN1GAAKMT2A
SCHEMBL20150816 0.76 GRIN2D (0.38) HPGDALDH1A1MAPTKDM4EMEN1
SCHEMBL1797414 0.76 VCAM1 (0.38) HPGDMAPTKDM4EMEN1KMT2A
SCHEMBL1797415 0.76 VCAM1 (0.38) HPGDMAPTKDM4EMEN1KMT2A
SCHEMBL7375104 0.76 GRIN2D (0.38) HPGDALDH1A1MAPTKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1151990-A1 Substituted N-arylmethylamino derivatives of cyclobutene-3, 4-diones AMERICAN HOME PRODUCTS CORPORATION (US) 2001-11-07 EP disclosed
EP-0934257-A1 SUBSTITUTED N-ARYLMETHYLAMINO DERIVATIVES OF CYCLOBUTENE-3,4-DIONES AMERICAN HOME PRODUCTS CORPORATION (US) 1999-08-11 EP disclosed
US-5780505-A ADMINISTERING AS SMOOTH MUSCLE RELAXANT AMERICAN HOME PRODUCTS CORPORATION (US) 1998-07-14 US disclosed
WO-1998002413-A1 SUBSTITUTED N-ARYLMETHYLAMINO DERIVATIVES OF CYCLOBUTENE-3,4-DIONES AMERICAN HOME PRODUCTS CORPORATION (US) 1998-01-22 WO disclosed