SCHEMBL789348

SCHEMBL789348

CCCNS(=O)(=O)c1ccc(C)cc1NCCS

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.40
CA12 O43570 2/20 0.40
CA9 Q16790 2/20 0.40
TDP1 Q9NUW8 1/20 0.39
METAP2 P50579 1/20 0.38
MEP1B Q16820 2/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
KMT2A Q03164 1/20 0.38
FBP1 P09467 1/20 0.36
ALDH1A1 P00352 2/20 0.36
ADRA2A P08913 1/20 0.36
ADRA2C P18825 1/20 0.36
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
BRD4 O60885 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL801417 0.74 TDP1 (0.62) POLBL3MBTL1TDP1KMT2AALDH1A1
SCHEMBL801402 0.72 POLB (0.52) POLBL3MBTL1CA12CA9TDP1
SCHEMBL16261330 0.71 CNR2 (0.50) POLBL3MBTL1CA12CA9KMT2A
SCHEMBL11570203 0.70 POLB (0.47) POLBL3MBTL1TDP1METAP2ALDH1A1
SCHEMBL10700475 0.69 POLB (0.63) POLBL3MBTL1KMT2AALDH1A1
SCHEMBL634316 0.67 ALDH1A1 (0.71) L3MBTL1CA12CA9CA1CA2
SCHEMBL27903070 0.66 CA12 (0.52) POLBL3MBTL1CA12CA9TDP1
SCHEMBL17798993 0.65 ALDH1A1 (0.69) L3MBTL1CA12CA9CA1CA2
SCHEMBL11707958 0.65 KMT2A (0.83) CA12CA9CA1CA2KMT2A
SCHEMBL9230028 0.65 CA12 (0.54) POLBL3MBTL1CA12CA9TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1437139-B1 Method for protection against genotoxic mutagenesis ARCH DEV CORP (US) 2008-07-16 EP claimed
EP-1437139-A2 Method for protection against genotoxic mutagenesis ARCH DEVELOPMENT CORPORATION (US) 2004-07-14 EP claimed
EP-0764027-A4 METHOD FOR PROTECTION AGAINST GENOTOXIC MUTAGENESIS ARCH DEV CORP (US) 1998-04-22 EP claimed
EP-0764027-A1 METHOD FOR PROTECTION AGAINST GENOTOXIC MUTAGENESIS ARCH DEVELOPMENT CORPORATION (US) 1997-03-26 EP claimed
US-5488042-A Method for protection against genotoxic mutagenesis ARCH DEVELOPMENT CORPORATION (US) 1996-01-30 US claimed
WO-1995007700-A1 METHOD FOR PROTECTION AGAINST GENOTOXIC MUTAGENESIS ARCH DEVELOPMENT CORPORATION (US) 1995-03-23 WO claimed
WO-1993017689-A1 METHOD FOR PROTECTION AGAINST GENOTOXIC MUTAGENESIS ARCH DEVELOPMENT CORPORATION (US) 1993-09-16 WO claimed
EP-3632419-B1 METHODS AND COMPOSITIONS FOR PROTECTION OF CELLS AND TISSUES FROM COMPUTED TOMOGRAPHY RADIATION UNIV CHICAGO (US) 2022-12-28 EP disclosed
US-20210244751-A1 METHODS AND COMPOSITIONS FOR PROTECTION OF CELLS AND TISSUES FROM COMPUTED TOMOGRAPHY RADIATION THE UNIVERSITY OF CHICAGO (US) 2021-08-12 US disclosed
EP-3632419-A1 METHODS AND COMPOSITIONS FOR PROTECTION OF CELLS AND TISSUES FROM COMPUTED TOMOGRAPHY RADIATION The University of Chicago (US) 2020-04-08 EP disclosed
US-20150231093-A1 METHODS AND COMPOSITIONS FOR COUNTERMEASURES AGAINST RADIATION NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2015-08-20 US disclosed
EP-2663297-A2 METHODS AND COMPOSITIONS FOR PROTECTION OF CELLS AND TISSUES FROM COMPUTED TOMOGRAPHY RADIATION The University of Chicago (US) 2013-11-20 EP disclosed
WO-2012037466-A2 METHODS AND COMPOSITIONS FOR PROTECTION CELLS AND TISSUES FROM COMPUTED TOMOGRAPHY RADIATION THE UNIVERSITY OF CHICAGO (US) 2012-03-22 WO disclosed
EP-1437139-A2 Method for protection against genotoxic mutagenesis ARCH DEVELOPMENT CORPORATION (US) 2004-07-14 EP disclosed
US-5869338-A Method for protection against genotoxic mutagenesis ARCH DEVELOPMENT CORPORATION (US) 1999-02-09 US disclosed
EP-0764027-A4 METHOD FOR PROTECTION AGAINST GENOTOXIC MUTAGENESIS ARCH DEV CORP (US) 1998-04-22 EP disclosed
EP-0764027-A1 METHOD FOR PROTECTION AGAINST GENOTOXIC MUTAGENESIS ARCH DEVELOPMENT CORPORATION (US) 1997-03-26 EP disclosed
US-5488042-A Method for protection against genotoxic mutagenesis ARCH DEVELOPMENT CORPORATION (US) 1996-01-30 US disclosed
WO-1995007700-A1 METHOD FOR PROTECTION AGAINST GENOTOXIC MUTAGENESIS ARCH DEVELOPMENT CORPORATION (US) 1995-03-23 WO disclosed
WO-1993017689-A1 METHOD FOR PROTECTION AGAINST GENOTOXIC MUTAGENESIS ARCH DEVELOPMENT CORPORATION (US) 1993-09-16 WO disclosed